SCHEMBL8729916

SCHEMBL8729916

O=C1Cn2c(nc3ccccc32)NN1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.46
KDM4E B2RXH2 6/20 0.41
HSD17B10 Q99714 3/20 0.41
NPC1 O15118 1/20 0.41
TP53 P04637 1/20 0.41
PKM P14618 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
ALDH1A1 P00352 7/20 0.39
HPGD P15428 5/20 0.39
IRAK4 Q9NWZ3 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ZAP70 P43403 1/20 0.37
POLB P06746 1/20 0.37
MAPT P10636 2/20 0.37
LMNA P02545 1/20 0.37
GRM2 Q14416 1/20 0.37
GLA P06280 1/20 0.37
HTT P42858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1699146 0.85 TSHR (0.47) TSHRKDM4EHSD17B10NPC1TP53
SCHEMBL1713613 0.72 CRBN (0.44) TSHRKDM4EHSD17B10ALDH1A1HPGD
SCHEMBL32688313 0.72 CRBN (0.44) TSHRKDM4EHSD17B10ALDH1A1HPGD
SCHEMBL839645 0.67 KDM4E (0.61) TSHRKDM4EHSD17B10NPC1TP53
SCHEMBL14974497 0.67 KDM4E (0.41) TSHRKDM4EHSD17B10NPC1TP53
SCHEMBL31249024 0.67 KDM4E (0.61) TSHRKDM4EHSD17B10NPC1TP53
SCHEMBL1713450 0.66 TSHR (0.42) TSHRKDM4ESMN1; SMN2ALDH1A1HPGD
SCHEMBL5142126 0.66 ALDH1A1 (0.47) TSHRKDM4EHSD17B10RAB9ASMN1; SMN2
SCHEMBL8797169 0.65 ALPI (0.41) TSHRKDM4ESMN1; SMN2ALDH1A1HPGD
SCHEMBL840080 0.64 KDM4E (0.63) TSHRKDM4EHSD17B10NPC1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998043649-A2 AGE PRODUCTION INHIBITORY COMPOSITION COMPRISING A MAILLARD REACTION INHIBITOR AND VITAMIN B¿6? OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-10-08 WO disclosed