SCHEMBL8733429

SCHEMBL8733429

O=C(O)Oc1cn(C2CC2)c2c(Cl)c(F)ccc2c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
POLB P06746 2/20 0.43
OPRM1 P35372 2/20 0.43
CHRM2 P08172 1/20 0.43
CHRM1 P11229 1/20 0.43
OPRD1 P41143 1/20 0.43
TOP2A P11388 6/20 0.40
TOP2B Q02880 6/20 0.40
KCNH2 Q12809 5/20 0.35
GSK3B P49841 2/20 0.35
PIK3CD O00329 1/20 0.35
PIK3R1 P27986 1/20 0.35
PIK3CA P42336 1/20 0.35
PIK3CG P48736 1/20 0.35
KDM4E B2RXH2 1/20 0.34
PRKD3 O94806 1/20 0.34
HPGD P15428 1/20 0.34
ALOX15 P16050 1/20 0.34
CLK2 P49760 1/20 0.34
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9044178 0.88 TOP2A (0.47) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL9416398 0.86 CYP3A4 (0.39) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL9416381 0.86 CYP3A4 (0.39) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL9416477 0.86 CYP3A4 (0.39) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL9416458 0.86 KCNH2 (0.41) ALDH1A1POLBOPRM1TOP2ATOP2B
SCHEMBL10915183 0.86 TOP2A (0.43) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL1972628 0.85 ALDH1A1 (0.49) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL4482132 0.84 ALDH1A1 (0.58) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL9416470 0.84 KCNH2 (0.46) ALDH1A1POLBOPRM1TOP2ATOP2B
SCHEMBL8785244 0.84 TOP2A (0.39) ALDH1A1POLBOPRM1CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0607825-A1 6-H-4-OXO-3-quinoline-carboxylic acids and their analogues as antibacterial agents BAYER AG (DE) 1994-07-27 EP claimed
EP-0607824-B1 Method for the production of multiply halogenated benzotrichlorides and benzoyl chlorides as well as new multiply halogenated benzotrichlorides BAYER AG (DE) 1998-04-22 EP disclosed
EP-0588166-B1 Antibacterial 7-isoindolinyl-quinolone and naphthyridone derivatives BAYER AG (DE) 1996-06-05 EP disclosed
EP-0607824-A2 Method for the production of multiply halogenated benzotrifluorides, benzotrichlorides and benzoyl chlorides as well as trihalobenzotrichlorides and -benzoyl chlorides BAYER AG (DE) 1994-07-27 EP disclosed
EP-0607825-A1 6-H-4-OXO-3-quinoline-carboxylic acids and their analogues as antibacterial agents BAYER AG (DE) 1994-07-27 EP disclosed
EP-0588166-A2 Antibacterial 7-isoindolinyl-quinolone and naphthyridone derivatives BAYER AG (DE) 1994-03-23 EP disclosed