SCHEMBL8733651

SCHEMBL8733651

COc1ccc(-c2sc3ccccc3c2C(=O)c2ccc(OCCN(C(C)C)C(C)C)cc2)cc1.COc1ccc(-c2sc3ccccc3c2C(=O)c2ccc(OCCN(C)C)cc2)cc1

nearest known ligand 0.66

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 5/20 0.66
CNR1 P21554 3/20 0.66
PAX8 Q06710 1/20 0.62
ESR1 P03372 10/20 0.61
ESR2 Q92731 10/20 0.61
ITGA4 P13612 1/20 0.55
NAPEPLD Q6IQ20 1/20 0.55
ATM Q13315 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
ENPP3 O14638 1/20 0.49
ENPP1 P22413 1/20 0.49
HCRTR1 O43613 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4651853 0.96 CNR2 (0.71) CNR2CNR1PAX8ESR1ESR2
SCHEMBL4652009 0.93 CNR2 (0.75) CNR2CNR1PAX8ESR1ESR2
SCHEMBL11550720 0.89 CNR1 (0.67) CNR2CNR1PAX8ESR1ESR2
SCHEMBL4651997 0.89 ESR1 (0.64) CNR2CNR1ESR1ESR2TDP1
SCHEMBL11547037 0.86 CNR1 (0.62) CNR2CNR1PAX8ESR1ESR2
SCHEMBL11545740 0.86 ESR1 (0.67) CNR2CNR1PAX8ESR1ESR2
SCHEMBL4651840 0.86 ESR1 (0.67) CNR2CNR1PAX8ESR1ESR2
SCHEMBL11555855 0.85 ESR1 (0.68) CNR2CNR1PAX8ESR1ESR2
SCHEMBL4650716 0.84 CNR2 (0.72) CNR2CNR1PAX8ESR1ESR2
SCHEMBL11550741 0.84 CNR2 (0.72) CNR2CNR1PAX8ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0820769-A2 Use of benzothiophenes for the manufacture of a medicament for the treatment of diseases associated with an excess of tachykinis ELI LILLY AND COMPANY (US) 1998-01-28 EP claimed