SCHEMBL11550720

SCHEMBL11550720

CN(C)CCOc1ccc(C(=O)c2c(-c3ccc(OCCN(C)C)cc3)sc3ccccc23)cc1

nearest known ligand 0.67

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 2/20 0.67
CNR2 P34972 2/20 0.67
PAX8 Q06710 1/20 0.62
ESR1 P03372 12/20 0.62
ESR2 Q92731 12/20 0.62
ITGA4 P13612 1/20 0.57
NAPEPLD Q6IQ20 1/20 0.57
F2 P00734 1/20 0.55
ATM Q13315 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
HCRTR1 O43613 1/20 0.50
ENPP1 P22413 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11547037 0.97 CNR1 (0.62) CNR1CNR2PAX8ESR1ESR2
SCHEMBL11545740 0.96 ESR1 (0.67) CNR1CNR2PAX8ESR1ESR2
SCHEMBL4652009 0.96 CNR2 (0.75) CNR1CNR2PAX8ESR1ESR2
SCHEMBL4651840 0.96 ESR1 (0.67) CNR1CNR2PAX8ESR1ESR2
SCHEMBL8733651 0.89 CNR2 (0.66) CNR1CNR2PAX8ESR1ESR2
SCHEMBL6595454 0.89 ESR1 (0.80) CNR1ESR1ESR2F2TDP1
SCHEMBL11548759 0.87 ESR1 (0.66) CNR1CNR2PAX8ESR1ESR2
SCHEMBL11555273 0.87 ESR1 (0.66) CNR1ESR1ESR2TDP1
SCHEMBL8596134 0.86 ESR1 (0.60) CNR1CNR2PAX8ESR1ESR2
SCHEMBL11546663 0.86 ESR1 (0.62) CNR1ESR1ESR2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4133814-A ANTITUMOR AGENTS ELI LILLY AND COMPANY (US) 1979-01-09 US disclosed