SCHEMBL8734246

SCHEMBL8734246

COC(=O)c1ccc(C(C)C#N)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.50
CA2 P00918 3/20 0.50
CA12 O43570 2/20 0.50
CA9 Q16790 2/20 0.50
CA14 Q9ULX7 2/20 0.50
TDP1 Q9NUW8 1/20 0.50
CA7 P43166 1/20 0.50
TSHR P16473 1/20 0.47
MAPT P10636 6/20 0.46
ALDH1A1 P00352 3/20 0.46
KMT2A Q03164 3/20 0.45
MITF O75030 1/20 0.45
LMNA P02545 1/20 0.45
TP53 P04637 1/20 0.45
MAPK1 P28482 1/20 0.45
HTT P42858 1/20 0.45
RAPGEF3 O95398 1/20 0.45
RAB9A P51151 3/20 0.44
LOXL2 Q9Y4K0 1/20 0.44
NPC1 O15118 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31386185 1.00 CA1 (0.50) CA1CA2CA12CA9CA14
SCHEMBL3014304 0.83 CA1 (0.47) CA1CA2CA12CA9CA14
SCHEMBL23199299 0.81 MAPT (0.49) CA1CA2CA12CA9CA14
SCHEMBL14487928 0.81 CA1 (0.48) CA1CA2CA12CA9CA14
SCHEMBL2522006 0.80 LOXL2 (0.46) TSHRMAPTALDH1A1KMT2ATP53
SCHEMBL7302128 0.79 TSHR (0.48) CA1CA2CA12CA9CA14
SCHEMBL84424 0.79 CA1 (0.59) CA1CA2CA12CA9CA14
Cyanate SCHEMBL28803587 0.78 CA1 (0.64) CA1CA2CA12CA9CA14
SCHEMBL20504196 0.78 MAPT (0.46) CA1CA2CA12CA9CA14
Water SCHEMBL22720573 0.78 CA1 (0.76) CA1CA2CA12CA9CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117659022-A Ureido substituted pyridine compound, pharmaceutical composition containing ureido substituted pyridine compound and medical application of ureido substituted pyridine compound 苏州阿尔脉生物科技有限公司 2024-03-08 CN disclosed
WO-2022128850-A1 NOVEL ISOQUINOLINE DERIVATIVES AND PHARMACEUTICAL COPOSITIONS THEREOF FOR THE TREATMENT OF DISEASES GALAPAGOS NV (BE) 2022-06-23 WO disclosed
EP-0874826-A1 NAPHTHALENE QUINOLINES HAVING LEUKOTRIENE-ANTAGONISTIC ACTION LABORATORIOS MENARINI S.A. (ES) 1998-11-04 EP disclosed
WO-1997024331-A1 NAPHTHALENE QUINOLINES HAVING LEUKOTRIENE-ANTAGONISTIC ACTION LABORATORIOS MENARINI S.A. (ES) 1997-07-10 WO disclosed
CN-1094035-A Carboxylic acid derivative contains pharmaceutical composition of these compounds and preparation method thereof THOMAE GMBH DR K (DE) 1994-10-26 CN disclosed
EP-0604800-A1 4- 4- 4-(carboxyalkyl)-phenyl amino carbonyl -phenyl -piperedines as aggregation inhibitors Dr. Karl Thomae GmbH (DE) 1994-07-06 EP disclosed
US-5135949-A Anticoagulants BOEHRINGER MANNHEIM GMBH (DE) 1992-08-04 US disclosed