Malonic Acid

Malonic Acid

SCHEMBL8735862

C=CCOC(=O)C=C.O=C(O)CC(=O)O

nearest known ligand 0.48

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Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.48
CACNA1B Q00975 1/20 0.48
APBA1 Q02410 1/20 0.48
TSHR P16473 9/20 0.45
ALDH1A1 P00352 5/20 0.45
TP53 P04637 3/20 0.45
HIF1A Q16665 3/20 0.45
CYP3A4 P08684 3/20 0.45
HSD17B10 Q99714 3/20 0.45
SMN1; SMN2 Q16637 2/20 0.41
MAPK1 P28482 1/20 0.41
HPGD P15428 1/20 0.41
LDHA P00338 1/20 0.39
SRR Q9GZT4 1/20 0.39
ALOX15 P16050 1/20 0.39
THRB P10828 2/20 0.38
APP P05067 1/20 0.37
TDP1 Q9NUW8 1/20 0.33
PKM P14618 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL1577827 0.89 TSHR (0.50) MAPTCACNA1BAPBA1TSHRALDH1A1
SCHEMBL5167665 0.89 TSHR (0.54) MAPTCACNA1BAPBA1TSHRALDH1A1
SCHEMBL31267242 0.89 TSHR (0.54) MAPTCACNA1BAPBA1TSHRALDH1A1
SCHEMBL19273 0.89
Itaconate SCHEMBL2641437 0.87 HSD17B10 (0.60) MAPTCACNA1BAPBA1TSHRALDH1A1
Acrylic Acid SCHEMBL28462478 0.86 TSHR (0.48) MAPTCACNA1BAPBA1TSHRALDH1A1
Acrylic Acid SCHEMBL170500 0.86 TSHR (0.48) MAPTCACNA1BAPBA1TSHRALDH1A1
Charcoal, Activated SCHEMBL3744730 0.86
Water SCHEMBL1079113 0.86
Ethylene SCHEMBL5184263 0.86 TSHR (0.52) MAPTCACNA1BAPBA1TSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0735998-B1 PROCESS FOR PREPARING MICHAEL ADDITION PRODUCTS ALBEMARLE CORP (US) 1998-10-14 EP disclosed
EP-0735998-B1 PROCESS FOR PREPARING MICHAEL ADDITION PRODUCTS ALBEMARLE CORP (US) 1998-10-14 EP disclosed
US-5648018-A Ester/polyolefin refrigeration lubricant ALBEMARLE CORPORATION (US) 1997-07-15 US disclosed
EP-0735998-A1 PROCESS FOR PREPARING MICHAEL ADDITION PRODUCTS ALBEMARLE CORPORATION (US) 1996-10-09 EP disclosed
EP-0735998-A1 PROCESS FOR PREPARING MICHAEL ADDITION PRODUCTS ALBEMARLE CORPORATION (US) 1996-10-09 EP disclosed
WO-1995017368-A1 PROCESS FOR PREPARING MICHAEL ADDITION PRODUCTS ALBEMARLE CORPORATION (US) 1995-06-29 WO disclosed
WO-1995017368-A1 PROCESS FOR PREPARING MICHAEL ADDITION PRODUCTS ALBEMARLE CORPORATION (US) 1995-06-29 WO disclosed
US-5347043-A REACTING A DIALKYL MALONATE WITH AT LEAST THREE MOLAR PROPORTIONS OF AN ALKYL ACRYLATE IN THE PRESENCE OF A BASIC INITIATOR AND A PHASE TRANSFER CATALYST ALBEMARLE CORPORATION (US) 1994-09-13 US disclosed
US-5347043-A REACTING A DIALKYL MALONATE WITH AT LEAST THREE MOLAR PROPORTIONS OF AN ALKYL ACRYLATE IN THE PRESENCE OF A BASIC INITIATOR AND A PHASE TRANSFER CATALYST ALBEMARLE CORPORATION (US) 1994-09-13 US disclosed