SCHEMBL8737860

SCHEMBL8737860

C=C(C)C(CC#N)c1cc(OCC#N)ccc1C#N

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.34
GLA P06280 2/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH2 P05091 1/20 0.34
GAA P10253 1/20 0.34
HPGD P15428 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HSD17B10 Q99714 1/20 0.34
MAOB P27338 3/20 0.33
MAOA P21397 2/20 0.33
MAPT P10636 2/20 0.32
TSHR P16473 2/20 0.32
NPC1 O15118 2/20 0.32
RAB9A P51151 2/20 0.32
SLC2A1 P11166 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
MRGPRX4 Q96LA9 1/20 0.31
PSEN1 P49768 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL171678 0.80 ALDH1A1 (0.37) ALDH1A1GLAL3MBTL1KDM4EALDH2
SCHEMBL9918234 0.77 MAOB (0.37) ALDH1A1GLAL3MBTL1KDM4EALDH2
SCHEMBL19592355 0.76 ALDH1A1 (0.35) ALDH1A1GLAL3MBTL1KDM4EALDH2
SCHEMBL19592356 0.74 ALDH1A1 (0.34) ALDH1A1GLAL3MBTL1KDM4EALDH2
SCHEMBL9918862 0.72 MAOB (0.35) ALDH1A1GLAL3MBTL1KDM4EALDH2
SCHEMBL24595040 0.69 ALDH1A1 (0.40) ALDH1A1GLAL3MBTL1KDM4EALDH2
SCHEMBL16954255 0.66 GLA (0.46) ALDH1A1GLAL3MBTL1KDM4EGAA
SCHEMBL16957324 0.66 GLA (0.43) ALDH1A1GLAL3MBTL1KDM4EHPGD
SCHEMBL9921725 0.66 KDM4E (0.37) ALDH1A1GLAL3MBTL1KDM4EALDH2
SCHEMBL12041228 0.65 GLA (0.48) ALDH1A1GLAL3MBTL1KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2455382-A1 Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors Incyte Corporation (US) 2012-05-23 EP disclosed