SCHEMBL874002

SCHEMBL874002

COc1cccc2nn[nH]c(=O)c12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ELANE P08246 2/20 0.45
KDM4E B2RXH2 3/20 0.42
ALDH1A1 P00352 3/20 0.42
HPGD P15428 3/20 0.42
DCPS Q96C86 1/20 0.41
KEAP1 Q14145 1/20 0.41
NFE2L2 Q16236 1/20 0.41
ABCG2 Q9UNQ0 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
GAA P10253 1/20 0.39
MAPK1 P28482 1/20 0.39
HSD17B10 Q99714 1/20 0.39
MMP13 P45452 1/20 0.39
NQO2 P16083 1/20 0.39
PDE3B Q13370 1/20 0.38
PDE3A Q14432 1/20 0.38
POLB P06746 1/20 0.38
MAPT P10636 1/20 0.38
ALOX15 P16050 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10882640 0.77 PARP1 (0.54) ELANE
SCHEMBL18643654 0.75 PDE3B (0.50) KDM4EALDH1A1HPGDABCG2GAA
SCHEMBL11144420 0.75 KEAP1 (0.46) KDM4EALDH1A1HPGDDCPSKEAP1
SCHEMBL873756 0.74 PARP1 (0.54) MMP13POLB
SCHEMBL6610267 0.74 PARP1 (0.38) KDM4EALDH1A1HPGDKMT2AGAA
SCHEMBL17950745 0.74 PDPK1 (0.37) ALOX15
SCHEMBL17950543 0.74 PDPK1 (0.44) ELANEKMT2AGUSB
SCHEMBL28960473 0.74 AXL (0.44) KDM4EALDH1A1MEN1KMT2AHSD17B10
SCHEMBL874607 0.74 PARP1 (0.54) ELANEGAAGUSB
SCHEMBL873985 0.73 TNKS (0.51) KDM4EALDH1A1HPGDKEAP1NFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016116058-A1 TRIAZINE HETEROCYCLIC COMPOUND WITH NEMATICIDAL ACTIVITY AND PREPARATION METHOD THEREFOR AND USAGE THEREOF 华东理工大学 2016-07-28 WO disclosed
EP-2619179-A1 MATRIX METALLOPROTEINASE INHIBITORS Ranbaxy Laboratories Limited (IN) 2013-07-31 EP disclosed
WO-2012038944-A1 MATRIX METALLOPROTEINASE INHIBITORS RANBAXY LABORATORIES LIMITED (IN) 2012-03-29 WO disclosed