SCHEMBL8740097

SCHEMBL8740097

N#Cc1ccc(-c2nc3ccc(O)cc3o2)cc1

nearest known ligand 0.74

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 13/20 0.74
ESR2 Q92731 13/20 0.74
NPC1 O15118 1/20 0.58
RAB9A P51151 1/20 0.58
HDAC6 Q9UBN7 1/20 0.53
GPR119 Q8TDV5 1/20 0.51
APP P05067 3/20 0.50
CYP19A1 P11511 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5031906 0.88 ESR1 (0.74) ESR1ESR2HDAC6APP
SCHEMBL27090228 0.87 ESR1 (0.96) ESR1ESR2NPC1RAB9AAPP
SCHEMBL2158317 0.86 ESR1 (1.00) ESR1ESR2NPC1RAB9AAPP
SCHEMBL24038264 0.81 ESR1 (0.51) ESR1ESR2NPC1RAB9AHDAC6
SCHEMBL2248809 0.80 ESR1 (0.81) ESR1ESR2NPC1RAB9AAPP
SCHEMBL17561646 0.80 ESR1 (0.81) ESR1ESR2NPC1RAB9A
SCHEMBL9114641 0.80 ESR1 (0.81) ESR1ESR2NPC1RAB9AHDAC6
SCHEMBL16894055 0.80 ESR1 (0.81) ESR1ESR2NPC1RAB9AAPP
SCHEMBL31278592 0.80 GPR119 (0.52) ESR1ESR2NPC1RAB9AHDAC6
SCHEMBL8034090 0.80 ESR1 (0.81) ESR1ESR2NPC1RAB9AAPP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5696001-A DETECTION OF HYDROLASES BEHRINGWERKE AKTIENGESELLSCHAFT (DE) 1997-12-09 US disclosed
US-5648229-A DETECTION OF HYDROLYTIC ENZYMES BEHRINGWERKE AKTIENGESELLSCHAFT (DE) 1997-07-15 US disclosed
US-5585247-A FLUORESCENT DYES FOR ENZYME IMMUNOASSAY BEHRINGWERKE AKTIENGESELLSCHAFT (DE) 1996-12-17 US disclosed
EP-0399409-A2 Fluorogene compounds and their use BEHRINGWERKE Aktiengesellschaft (DE) 1990-11-28 EP disclosed