SCHEMBL8742149

SCHEMBL8742149

CCNc1cc(Cl)cc(C(=O)O)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TPMT P51580 1/20 0.55
HCAR1 Q9BXC0 1/20 0.48
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
GAA P10253 3/20 0.42
ALDH1A1 P00352 2/20 0.42
MAPT P10636 2/20 0.42
KDM4E B2RXH2 1/20 0.42
THRB P10828 1/20 0.42
HPGD P15428 1/20 0.42
HTT P42858 1/20 0.42
GFER P55789 1/20 0.42
PLEC Q15149 1/20 0.42
WDR5 P61964 2/20 0.42
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
IDO1 P14902 1/20 0.41
TDO2 P48775 1/20 0.41
FABP4 P15090 1/20 0.40
HCAR3 P49019 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7076066 0.87 MEN1 (0.50) TPMTMEN1KMT2AGAAALDH1A1
SCHEMBL14107722 0.79 TPMT (0.61) TPMTHCAR1MEN1KMT2AALDH1A1
SCHEMBL3398764 0.78 ALDH1A1 (0.42) GAAALDH1A1MAPTKDM4EHPGD
SCHEMBL3793129 0.78 EGFR (0.40) GAAALDH1A1MAPTKDM4EHPGD
SCHEMBL27620238 0.77 KDM4E (0.53) MEN1KMT2AGAAALDH1A1MAPT
SCHEMBL8742132 0.77 PPARA (0.57) TPMTMEN1KMT2AALDH1A1MAPT
Hydrochloric Acid SCHEMBL8956072 0.77 HTR2B (0.42)
Hydrochloric Acid SCHEMBL3396163 0.76 ALDH1A1 (0.41) GAAALDH1A1MAPTKDM4EHPGD
Hydrochloric Acid SCHEMBL8742155 0.76 ALDH1A1 (0.35) GAAALDH1A1MAPTHPGDNPC1
SCHEMBL28582621 0.75 TPMT (0.55) TPMTHCAR1MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0603650-B1 3,5-Substituted amino benzoylguanidines, process for their preparation, their use as medicine or diagnostic agent, as well as a medicine containing them HOECHST AG (DE) 1997-04-02 EP disclosed
US-5516805-A 3,5-substituted aminobenzoylguanidines, their use as a medicament or diagnostic and medicament containing them HOECHST AKTIENGESELLSCHAFT (DE) 1996-05-14 US disclosed
EP-0603650-A1 3,5-Substituted amino benzoylguanidines, process for their preparation, their use as medicine or diagnostic agent, as well as a medicine containing them HOECHST AKTIENGESELLSCHAFT (DE) 1994-06-29 EP disclosed