SCHEMBL8742452

SCHEMBL8742452

CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](CO)Cc1c[nH]c2ccccc12

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSL P07711 2/20 0.66
CTSS P25774 1/20 0.66
CTSK P43235 1/20 0.66
ACE P12821 1/20 0.65
HDAC3 O15379 3/20 0.62
HDAC4 P56524 3/20 0.62
HDAC1 Q13547 3/20 0.62
HDAC7 Q8WUI4 3/20 0.62
HDAC2 Q92769 3/20 0.62
HDAC10 Q969S8 3/20 0.62
HDAC11 Q96DB2 3/20 0.62
HDAC8 Q9BY41 3/20 0.62
HDAC6 Q9UBN7 3/20 0.62
HDAC9 Q9UKV0 3/20 0.62
HDAC5 Q9UQL6 3/20 0.62
MAPT P10636 2/20 0.61
TP53 P04637 1/20 0.61
CCKBR P32239 6/20 0.59
REN P00797 1/20 0.59
SMN1; SMN2 Q16637 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30638855 0.89 ACE (0.78) CTSLCTSSCTSKACEMAPT
SCHEMBL27885190 0.89 ACE (0.78) CTSLCTSSCTSKACEMAPT
SCHEMBL27885189 0.89 ACE (0.78) CTSLCTSSCTSKACEMAPT
SCHEMBL3825352 0.89 ACE (0.78) CTSLCTSSCTSKACEMAPT
SCHEMBL31484559 0.89 ACE (0.78) CTSLCTSSCTSKACEMAPT
SCHEMBL29401065 0.88 CTSL (0.63) CTSLCTSSCTSKACEHDAC3
SCHEMBL29398124 0.88 CTSL (0.63) CTSLCTSSCTSKACEHDAC3
SCHEMBL3560147 0.88 CTSL (0.63) CTSLCTSSCTSKACEHDAC3
SCHEMBL6409052 0.88 CTSL (0.63) CTSLCTSSCTSKACEHDAC3
SCHEMBL6833548 0.88 CTSL (0.63) CTSLCTSSCTSKACEHDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0783489-A1 ALDEHYDE DERIVATIVES AS UPSTEINE PROTEASE INHIBITORS Takeda Chemical Industries, Ltd. (JP) 1997-07-16 EP disclosed
WO-1996010014-A1 ALDEHYDE DERIVATIVES AS UPSTEINE PROTEASE INHIBITORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-04-04 WO disclosed