SCHEMBL8743553

SCHEMBL8743553

OCC(F)(F)CCOCc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.50
POLB P06746 1/20 0.50
TSHR P16473 1/20 0.48
PTPN2 P17706 1/20 0.41
PTPN1 P18031 1/20 0.41
PTPN6 P29350 1/20 0.41
CA1 P00915 1/20 0.41
CHRM3 P20309 4/20 0.40
CHRM2 P08172 2/20 0.40
CHRM1 P11229 2/20 0.40
SLC6A2 P23975 1/20 0.40
PDE4A P27815 1/20 0.40
SLC6A4 P31645 1/20 0.40
OPRM1 P35372 1/20 0.40
SLC6A3 Q01959 1/20 0.40
UGCG Q16739 2/20 0.39
GBA2 Q9HCG7 2/20 0.39
GBA1 P04062 1/20 0.39
SI P14410 1/20 0.39
NAAA Q02083 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21068792 0.88 TSHR (0.47) KDM4EPOLBTSHRPTPN2PTPN1
SCHEMBL21068743 0.86 TSHR (0.45) KDM4EPOLBTSHRPTPN2PTPN1
SCHEMBL9237332 0.86 KDM4E (0.50) KDM4EPOLBTSHRPTPN2PTPN1
SCHEMBL30782112 0.83 KDM4E (0.47) KDM4EPOLBTSHRPTPN2PTPN1
SCHEMBL9836818 0.82 TSHR (0.48) KDM4EPOLBTSHRPTPN2PTPN1
SCHEMBL8352025 0.81 KDM4E (0.53) KDM4EPOLBTSHRCA1CHRM3
SCHEMBL9241218 0.81 KDM4E (0.53) KDM4EPOLBTSHRCA1CHRM3
SCHEMBL9276198 0.81 KDM4E (0.62) KDM4EPOLBTSHRCA1UGCG
SCHEMBL21068524 0.81 KDM4E (0.50) KDM4EPOLBTSHRPTPN2PTPN1
SCHEMBL28776126 0.81 TSHR (0.56) KDM4EPOLBTSHRPTPN2PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0335770-B1 Novel fluorophosphonate nucleotide derivatives MERRELL PHARMA INC (US) 1997-01-15 EP disclosed
EP-0215319-B1 GEM-DIHALO-1,8-DIAMINO-4-AZA-OCTANES MERRELL DOW PHARMACEUTICALS INC. (US) 1991-10-16 EP disclosed
US-4914240-A PROTECTING DIHALO BUTANEDIOL, REACTING WITH POTASSIUM PHTHALIMINDE, DEPROTECTING; MULTISTEP MERRELL DOW PHARMACEUTICALS INC. (US) 1990-04-03 US disclosed
EP-0339161-A1 Novel fluorophosphonate nucleotide derivatives MERRELL DOW PHARMACEUTICALS INC. (US) 1989-11-02 EP disclosed
EP-0335770-A2 Novel fluorophosphonate nucleotide derivatives MERRELL PHARMACEUTICALS INC. (US) 1989-10-04 EP disclosed
US-4851448-A Gem-dihalo-1,8-diamino-4-aza-octanes MERRELL DOW PHARMACEUTICALS INC. (US) 1989-07-25 US disclosed
US-4695654-A ANTITUMOR AGENTS MERRELL DOW PHARMACEUTICALS INC. (US) 1987-09-22 US disclosed
EP-0215319-A2 Gem-dihalo-1,8-diamino-4-aza-octanes MERRELL DOW PHARMACEUTICALS INC. (US) 1987-03-25 EP disclosed