SCHEMBL8744339

SCHEMBL8744339

[CH2]C(C)Oc1ccc(C(F)(F)F)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.44
CYP3A5 P20815 1/20 0.44
SLC6A4 P31645 5/20 0.43
SLC6A2 P23975 4/20 0.43
SLC6A3 Q01959 4/20 0.43
MEN1 O00255 4/20 0.43
KMT2A Q03164 4/20 0.43
LMNA P02545 4/20 0.43
HRH3 Q9Y5N1 2/20 0.43
NPC1 O15118 2/20 0.43
CYP2D6 P10635 2/20 0.43
CYP2C19 P33261 2/20 0.43
MTOR P42345 2/20 0.43
RAB9A P51151 2/20 0.43
KCNK2 O95069 2/20 0.43
KCNH2 Q12809 2/20 0.43
CACNA1C Q13936 2/20 0.43
HTR2C P28335 2/20 0.43
KDM4E B2RXH2 1/20 0.43
TP53 P04637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL178405 0.83 CYP3A4 (0.58) CYP3A4CYP3A5SLC6A4SLC6A2SLC6A3
SCHEMBL15473214 0.76 SLC6A4 (0.44) CYP3A4CYP3A5SLC6A4SLC6A2SLC6A3
SCHEMBL11611228 0.76 SLC6A4 (0.44) CYP3A4CYP3A5SLC6A4SLC6A2SLC6A3
SCHEMBL11515859 0.76 CYP3A4 (0.40) CYP3A4CYP3A5SLC6A4SLC6A2SLC6A3
SCHEMBL20563547 0.76 PPARG (0.49) CYP3A4SLC6A4SLC6A2SLC6A3MEN1
SCHEMBL3165936 0.76 ALDH1A1 (0.47) SLC6A4MEN1KMT2ALMNAACHE
SCHEMBL25215833 0.75 PPARG (0.42) CYP3A4CYP3A5SLC6A4SLC6A2SLC6A3
SCHEMBL18071748 0.75 SLC6A4 (0.43) CYP3A4CYP3A5SLC6A4SLC6A2SLC6A3
SCHEMBL22809555 0.75 SLC6A4 (0.50) CYP3A4SLC6A4SLC6A2SLC6A3MEN1
SCHEMBL8888174 0.75 PPARG (0.42) CYP3A4CYP3A5SLC6A4SLC6A2SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691340-A CENTRAL NERVOUS SYSTEM DISORDERS, STROKES, CARDIOVASCULAR DISORDERS, ALZHEIMER*S DISEASE OR ANTIINFLAMMATORY AGENTS ADIR ET COMPAGNIE (FR) 1997-11-25 US disclosed
EP-0599906-B1 HERBICIDES CONTAINING 3-AMINOBENZO B]THIOPHENES AS AN ANTIDOTE BASF AG (DE) 1997-01-15 EP disclosed
EP-0552493-B1 Thiochromenone derivatives as antidotes and herbicidal agents containing them BASF AG (DE) 1996-09-11 EP disclosed
US-5491123-A Herbicides containing 3-aminobenzo(B)thiophenes as antidotes BASF AKTIENGESELLSCHAFT (DE) 1996-02-13 US disclosed
US-5378677-A Applying with cyclohexenone derivative BASF AKTIENGESELLSCHAFT (DE) 1995-01-03 US disclosed
EP-0599906-A1 HERBICIDES CONTAINING 3-AMINOBENZO B]THIOPHENES AS AN ANTIDOTE. BASF AG (DE) 1994-06-08 EP disclosed
EP-0552493-A1 Thiochromenone derivatives as antidotes and herbicidal agents containing them BASF Aktiengesellschaft (DE) 1993-07-28 EP disclosed
WO-1993004057-A2 HERBICIDES CONTAINING 3-AMINOBENZO[B]THIOPHENES AS AN ANTIDOTE BASF AKTIENGESELLSCHAFT (DE) 1993-03-04 WO disclosed