SCHEMBL8744773

SCHEMBL8744773

Cc1[nH]c(C#N)nc1-c1ccncc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.44
PDE5A O76074 1/20 0.44
LMNA P02545 1/20 0.44
HPGD P15428 1/20 0.44
TSHR P16473 1/20 0.44
PTGS1 P23219 1/20 0.44
PDE4A P27815 1/20 0.44
CYP2C19 P33261 1/20 0.44
BLM P54132 1/20 0.44
PDE4B Q07343 1/20 0.44
PDE4C Q08493 1/20 0.44
PDE4D Q08499 1/20 0.44
PDE3B Q13370 1/20 0.44
PDE3A Q14432 1/20 0.44
ADORA1 P30542 2/20 0.41
ADORA2A P29274 1/20 0.41
MAPK14 Q16539 5/20 0.40
MAPK13 O15264 4/20 0.40
MAPK12 P53778 4/20 0.40
MAPK11 Q15759 4/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8744686 0.84 NPY5R (0.47) KDM4EHPGDTSHRADORA1ADORA2A
SCHEMBL8744702 0.84 ERBB2 (0.49) KDM4ELMNACYP2C19ADORA1ADORA2A
SCHEMBL30918737 0.73 MAPK14 (0.40) LMNAPDE3BPDE3AMAPK14MAPK13
SCHEMBL7300360 0.73 NPY5R (0.39) LMNAPDE3BPDE3AMAPK14MAPK13
SCHEMBL28399047 0.72 NPY5R (0.71) MAPK14MAPK13MAPK12MAPK11RAF1
SCHEMBL29330538 0.69 LRRK2 (0.50) KDM4EPDE5ALMNAHPGDTSHR
SCHEMBL21773988 0.68 ERBB2 (0.46) KDM4ELMNACYP2C19ADORA1ADORA2A
SCHEMBL8744781 0.66
SCHEMBL28402538 0.66 MAPK13 (0.63) MAPK14MAPK13MAPK12MAPK11RAF1
SCHEMBL7374799 0.65 SMPD3 (0.56) KDM4ELMNAHPGDMAPK14MAPK13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0653421-B1 Process for preparing 2-cyanoimidazole compounds ISHIHARA SANGYO KAISHA (JP) 1997-01-15 EP disclosed
US-5552557-A Process for preparing 2-cyanoimidazole compounds by reaction of an amino ketone compound ISHIHARA SANGYO KAISHA, LTD. (JP) 1996-09-03 US disclosed
EP-0653421-A1 Process for preparing 2-cyanoimidazole compounds ISHIHARA SANGYO KAISHA LTD. (JP) 1995-05-17 EP disclosed