Bicarbonate

Bicarbonate

SCHEMBL8744799

Cc1cc(C)c(CC(=O)NC2CC2)c(C)c1.O=C(O)O

nearest known ligand 0.49

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.49
TAS1R3 Q7RTX0 2/20 0.47
TAS1R1 Q7RTX1 2/20 0.47
TAS1R2 Q8TE23 2/20 0.47
EPHX2 P34913 2/20 0.46
LMNA P02545 2/20 0.46
HPGD P15428 1/20 0.46
SELL P14151 1/20 0.43
SELP P16109 1/20 0.43
SELE P16581 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL7615552 0.94 EPHX2 (0.46) KMT2ATAS1R3TAS1R1TAS1R2EPHX2
Bicarbonate SCHEMBL8744851 0.94 TAS1R3 (0.56) KMT2ATAS1R3TAS1R1TAS1R2EPHX2
Bicarbonate SCHEMBL8744732 0.92 TAS1R3 (0.59) KMT2ATAS1R3TAS1R1TAS1R2EPHX2
Bicarbonate SCHEMBL7615153 0.91 KMT2A (0.42) KMT2ATAS1R3TAS1R1TAS1R2EPHX2
Bicarbonate SCHEMBL7617866 0.90 KMT2A (0.41) KMT2ATAS1R3TAS1R1TAS1R2EPHX2
Bicarbonate SCHEMBL7622155 0.90 EPHX1 (0.43) KMT2ATAS1R3TAS1R1TAS1R2EPHX2
Bicarbonate SCHEMBL7614539 0.88 KMT2A (0.46) KMT2AEPHX2
Bicarbonate SCHEMBL7622402 0.87 KMT2A (0.38) KMT2ATAS1R3TAS1R1TAS1R2EPHX2
Bicarbonate SCHEMBL6996121 0.84 GAA (0.55) KMT2ATAS1R3TAS1R1TAS1R2EPHX2
Bicarbonate SCHEMBL6997216 0.83 NPC1 (0.54) KMT2ATAS1R3TAS1R1TAS1R2EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0456063-B1 1-H-3-aryl-pyrrolidin-2,4-dion-derivatives BAYER AG (DE) 1997-01-22 EP disclosed
EP-0456063-A2 1-H-3-aryl-pyrrolidin-2,4-dion-derivatives BAYER AG (DE) 1991-11-13 EP disclosed