SCHEMBL8745964

SCHEMBL8745964

CCc1ncncc1C(OC(=O)N(C)C)c1ccccc1C(F)(F)F

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 3/20 0.41
ITGA4 P13612 3/20 0.41
CYP3A4 P08684 4/20 0.35
TSHR P16473 3/20 0.35
KDM4E B2RXH2 3/20 0.35
HSD17B10 Q99714 2/20 0.35
TDP1 Q9NUW8 1/20 0.35
CYP2C19 P33261 3/20 0.35
CYP2D6 P10635 2/20 0.35
CYP1A2 P05177 2/20 0.35
KMT2A Q03164 1/20 0.34
POLQ O75417 1/20 0.33
ALDH1A1 P00352 1/20 0.33
ALOX15 P16050 1/20 0.33
MAPK1 P28482 1/20 0.33
CNR2 P34972 1/20 0.32
NEK2 P51955 2/20 0.32
PLK1 P53350 2/20 0.32
AURKA O14965 1/20 0.32
CDK2 P24941 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8745928 0.86 CYP3A4 (0.36) ITGB1ITGA4CYP3A4TSHRKDM4E
SCHEMBL8745942 0.85 CYP3A4 (0.37) ITGB1ITGA4CYP3A4TSHRKDM4E
SCHEMBL8745950 0.84 CYP3A4 (0.39) ITGB1ITGA4CYP3A4TSHRKDM4E
SCHEMBL9030025 0.78 GPBAR1 (0.38)
SCHEMBL8828275 0.77 CYP3A4 (0.39) CYP3A4TSHRKDM4EHSD17B10TDP1
SCHEMBL8326882 0.75 MAPT (0.40) POLQ
SCHEMBL8327868 0.74 MAPT (0.38) ITGB1ITGA4POLQ
SCHEMBL8745927 0.73 CCR4 (0.36) ITGB1ITGA4KMT2ACNR2NEK2
SCHEMBL8745915 0.73 CYP3A4 (0.39) ITGB1ITGA4CYP3A4TSHRKDM4E
SCHEMBL8549639 0.72 GPBAR1 (0.37) CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0758323-A1 HERBICIDAL HYDROXYBENZYL-SUBSTITUTED HETEROARYL COMPOUNDS AND DERIVATIVES THEREOF ZENECA LIMITED (GB) 1997-02-19 EP disclosed