SCHEMBL8747232

SCHEMBL8747232

CN1CCc2ccc(O)cc2C1C1(c2ccccc2Cl)CC1

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 12/20 0.45
HTR2A P28223 1/20 0.45
DRD2 P14416 7/20 0.45
DRD5 P21918 4/20 0.43
DRD3 P35462 3/20 0.43
DRD4 P21917 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL8747097 0.99 DRD1 (0.44) DRD1HTR2ADRD2DRD5DRD3
SCHEMBL8747078 0.95 DRD1 (0.44) DRD1HTR2ADRD2DRD5DRD3
Bromide SCHEMBL8747367 0.94 DRD1 (0.43) DRD1HTR2ADRD2DRD5DRD3
SCHEMBL8747024 0.85 DRD1 (0.47) DRD1DRD2DRD5DRD4
Hydrochloric Acid SCHEMBL8746990 0.84 DRD1 (0.46) DRD1DRD2DRD5DRD4
SCHEMBL8747039 0.84 DRD1 (0.46) DRD1DRD2DRD5DRD3DRD4
Bromide SCHEMBL8747087 0.84 DRD1 (0.46) DRD1DRD2DRD5DRD4
SCHEMBL8747331 0.83 DRD1 (0.44) DRD1DRD2DRD5DRD3DRD4
SCHEMBL8747167 0.83 MAOA (0.49) DRD1DRD2DRD5DRD3DRD4
Bromide SCHEMBL8747293 0.83 DRD1 (0.46) DRD1DRD2DRD5DRD3DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0618900-B1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS KNOLL AG (DE) 1997-03-12 EP disclosed
US-5519034-A ANALGESICS THE BOOTS COMPANY PLC (GB) 1996-05-21 US disclosed
EP-0618900-A1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS. BOOTS CO PLC (GB) 1994-10-12 EP disclosed
WO-1993013073-A1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS THE BOOTS COMPANY PLC (GB) 1993-07-08 WO disclosed