SCHEMBL8747233

SCHEMBL8747233

CN1CCc2cc(Br)c(O)cc2C1C1(c2ccccc2)CCC1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 10/20 0.52
DRD2 P14416 7/20 0.52
DRD5 P21918 3/20 0.52
CYP1A2 P05177 1/20 0.52
CYP2D6 P10635 1/20 0.52
TSHR P16473 1/20 0.52
CYP2C19 P33261 1/20 0.52
HSD17B10 Q99714 1/20 0.52
ADCY2 Q08462 1/20 0.52
LMNA P02545 1/20 0.51
ADRA2A P08913 1/20 0.51
ADRA2B P18089 1/20 0.51
ADRA2C P18825 1/20 0.51
SLC6A2 P23975 1/20 0.51
HTR1B P28222 1/20 0.51
HTR2A P28223 1/20 0.51
HTR2C P28335 1/20 0.51
MAPK1 P28482 1/20 0.51
SLC6A4 P31645 1/20 0.51
HTR7 P34969 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8747006 0.90 MAOA (0.50) DRD1DRD2HSD17B10MAPK1DRD3
Bromide SCHEMBL8747268 0.89 KDM4E (0.49) DRD1DRD2HSD17B10MAPK1DRD3
SCHEMBL8747355 0.88 MAOA (0.50) DRD1DRD2HSD17B10MAPK1DRD3
SCHEMBL8747054 0.87 MAOA (0.49) DRD1DRD2HSD17B10MAPK1DRD3
SCHEMBL8747056 0.86 DRD1 (0.60) DRD1DRD2DRD5CYP1A2CYP2D6
SCHEMBL8747186 0.86 DRD1 (0.43) DRD1DRD2DRD5HSD17B10MAPK1
SCHEMBL8747280 0.85 MAOA (0.52) DRD1DRD2HSD17B10MAPK1DRD3
SCHEMBL8747015 0.85 MAOA (0.47) DRD1DRD2DRD5HSD17B10MAPK1
SCHEMBL8747012 0.84 DRD1 (0.50) DRD1DRD2DRD5TSHRMAPK1
SCHEMBL8747360 0.84 MAOA (0.46) DRD1DRD2HSD17B10MAPK1DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0618900-B1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS KNOLL AG (DE) 1997-03-12 EP disclosed
WO-1993013073-A1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS THE BOOTS COMPANY PLC (GB) 1993-07-08 WO disclosed