SCHEMBL8747341

SCHEMBL8747341

COc1ccc2c(c1)C(C1(c3ccccc3Cl)CC1)=NCC2

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 2/20 0.40
MAPK10 P53779 3/20 0.39
MAOA P21397 2/20 0.39
LMNA P02545 2/20 0.38
MAPT P10636 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
SIGMAR1 Q99720 5/20 0.37
NPY5R Q15761 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA7 P43166 1/20 0.37
CA9 Q16790 1/20 0.37
CA14 Q9ULX7 1/20 0.37
MAOB P27338 1/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8747262 0.83 MAPT (0.45) MAPK14MAPK10MAOALMNAMAPT
SCHEMBL989662 0.82 SLC6A2 (0.49) LMNAMAPTNPSR1ALDH1A1
SCHEMBL8747316 0.82 MAPK10 (0.45) MAPK14MAPK10MAOALMNAMAPT
SCHEMBL8747277 0.80 NPY5R (0.43) MAPK14MAOAMAPTSIGMAR1NPY5R
SCHEMBL989046 0.78 SLC6A2 (0.47) MAOAMAPTMAOBALDH1A1
SCHEMBL8971786 0.77 MAPK10 (0.48) MAPK14MAPK10LMNAMAPTHTT
SCHEMBL8747185 0.77 KDM4E (0.48) MAPK14MAPK10LMNAMAPTHTT
SCHEMBL1862319 0.77 KDM4E (0.36) MAPK14MAPK10MAOAMAPTSIGMAR1
SCHEMBL7475657 0.76 NPY5R (0.43) MAPK14MAOAMAPTSIGMAR1NPY5R
SCHEMBL12629538 0.74 MAPT (0.41) MAOALMNAMAPTSMN1; SMN2NPY5R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0618900-B1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS KNOLL AG (DE) 1997-03-12 EP disclosed
US-5519034-A ANALGESICS THE BOOTS COMPANY PLC (GB) 1996-05-21 US disclosed
WO-1993013073-A1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS THE BOOTS COMPANY PLC (GB) 1993-07-08 WO disclosed