SCHEMBL8750928

SCHEMBL8750928

O=C(N[C@@H](Cc1ccccc1)C(=O)NC(O)C(=O)OCc1ccccc1)OCc1ccccc1

nearest known ligand 0.67

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 2/20 0.67
CTSL P07711 9/20 0.65
CTSB P07858 5/20 0.65
CTSS P25774 2/20 0.65
CTSK P43235 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8750885 0.92 CTSL (0.66) TACR1CTSLCTSBCTSSCTSK
SCHEMBL7295888 0.92 TACR1 (0.67) TACR1CTSLCTSBCTSSCTSK
SCHEMBL7269411 0.92 TACR1 (0.67) TACR1CTSLCTSBCTSSCTSK
SCHEMBL8668091 0.89 TACR1 (0.70) TACR1CTSLCTSBCTSSCTSK
SCHEMBL16095807 0.86 TACR1 (0.70) TACR1CTSLCTSBCTSSCTSK
SCHEMBL8100557 0.86 TACR1 (0.70) TACR1CTSLCTSBCTSSCTSK
SCHEMBL30688477 0.86 TACR1 (0.70) TACR1CTSLCTSBCTSSCTSK
SCHEMBL12052836 0.86 TACR1 (0.70) TACR1CTSLCTSBCTSSCTSK
SCHEMBL10049956 0.86 TACR1 (0.70) TACR1CTSLCTSBCTSSCTSK
SCHEMBL30241933 0.86 TACR1 (0.70) TACR1CTSLCTSBCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0561303-B1 Conjugates of phenylalanine-glycine with antitumor substances KUREHA CHEMICAL IND CO LTD (JP) 1997-02-26 EP disclosed
US-5470960-A Antitumor agents KUREHA CHEMICAL INDUSTRY CO., LTD. (JP) 1995-11-28 US disclosed
US-5411964-A Phenylalanine-glycine compounds having anti-tumor activity, process for preparation thereof, and pharmaceutical composition containing said compounds KUREHA CHEMICAL INDUSTRY CO., LTD. (JP) 1995-05-02 US disclosed