SCHEMBL8752010

SCHEMBL8752010

O=c1nc(C(F)(F)C(F)(F)F)cc[nH]1

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ELANE P08246 2/20 0.38
AXL P30530 1/20 0.31
NUDT1 P36639 1/20 0.31
PDE3B Q13370 1/20 0.31
PDE3A Q14432 1/20 0.31
DYRK1A Q13627 1/20 0.31
ADORA2A P29274 1/20 0.31
ADORA1 P30542 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2118961 0.83 FABP4 (0.37) ELANEAXLNUDT1
SCHEMBL8752056 0.76 ELANE (0.31) ELANE
SCHEMBL2355727 0.75 KDM4E (0.38) ELANEAXLNUDT1PDE3BPDE3A
SCHEMBL667243 0.69 JAK2 (0.33) ELANEDYRK1AADORA2AADORA1
SCHEMBL22627323 0.67 MAP2K1 (0.50) ELANE
SCHEMBL352936 0.67
Fluoride SCHEMBL31738503 0.67 DYRK1A (0.32) DYRK1AADORA2AADORA1
Fluoride SCHEMBL31738504 0.67 DYRK1A (0.32) DYRK1AADORA2AADORA1
SCHEMBL15496720 0.66 ELANE (0.32) ELANE
SCHEMBL1833402 0.66

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016113205-A1 SUBSTITUTED PENTAFLUOROETHYL PYRIMIDINONES AND USE THEREOF BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-07-21 WO disclosed
US-5684011-A Pyrimidine derivatives useful as nematicides ZENECA LIMITED (GB) 1997-11-04 US disclosed
EP-0660827-B1 HETEROCYCLIC COMPOUNDS WITH PARASITICAL ACTIVITY ZENECA LTD (GB) 1997-04-16 EP disclosed
WO-1994006777-A1 HETEROCYCLIC COMPOUNDS WIHT PARASITICAL ACTIVITY ZENECA LIMITED (GB) 1994-03-31 WO disclosed