SCHEMBL875389

SCHEMBL875389

Nc1ccc(-c2cc(N)c(C(=O)O)s2)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 6/20 0.60
CYP1A2 P05177 3/20 0.60
CYP2C9 P11712 3/20 0.60
CYP3A4 P08684 2/20 0.60
BTK Q06187 1/20 0.60
MAPT P10636 10/20 0.58
KDM4E B2RXH2 8/20 0.58
LMNA P02545 1/20 0.58
PKM P14618 1/20 0.58
RXFP1 Q9HBX9 1/20 0.58
CYP2C19 P33261 2/20 0.57
CHUK O15111 1/20 0.57
ALDH1A1 P00352 7/20 0.55
MEN1 O00255 6/20 0.55
KMT2A Q03164 6/20 0.55
POLB P06746 1/20 0.55
CDC7 O00311 1/20 0.53
DBF4 Q9UBU7 1/20 0.53
RAB9A P51151 6/20 0.53
GAA P10253 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29906389 0.89 IKBKB (0.60) IKBKBCYP1A2CYP2C9CYP3A4BTK
SCHEMBL2044907 0.87 IKBKB (0.77) IKBKBCYP1A2CYP2C9CYP3A4BTK
SCHEMBL3081896 0.86 MAPT (0.63) IKBKBCYP1A2CYP2C9CYP3A4BTK
SCHEMBL2313705 0.86 IKBKB (0.77) IKBKBCYP1A2CYP2C9CYP3A4BTK
SCHEMBL15881509 0.86 MAPT (0.59) IKBKBCYP1A2CYP2C9CYP3A4BTK
SCHEMBL1144476 0.86 IKBKB (0.77) IKBKBCYP1A2CYP2C9CYP3A4BTK
SCHEMBL2158576 0.86 IKBKB (0.75) IKBKBCYP1A2CYP2C9CYP3A4BTK
SCHEMBL6612593 0.86 IKBKB (0.76) IKBKBCYP1A2CYP2C9CYP3A4BTK
SCHEMBL4711452 0.85 PTPN1 (0.64) IKBKBCYP1A2CYP2C9CYP3A4BTK
SCHEMBL5193028 0.83 IKBKB (0.78) IKBKBCYP1A2CYP2C9CYP3A4BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012038904-A1 NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed