SCHEMBL875403

SCHEMBL875403

Nc1ccc(CNC(=O)Nc2ccc(-c3ccc(C(=O)NCCN4CCCCC4)o3)cc2)cn1

nearest known ligand 0.59

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 9/20 0.53
KIT P10721 1/20 0.47
HDAC1 Q13547 1/20 0.47
CHRM1 P11229 1/20 0.46
HTR2A P28223 1/20 0.46
MCHR1 Q99705 1/20 0.46
MEN1 O00255 1/20 0.44
POLB P06746 1/20 0.44
KMT2A Q03164 1/20 0.44
CNR1 P21554 1/20 0.44
ALDH1A1 P00352 1/20 0.43
ATR Q13535 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL875550 0.87 NAMPT (0.50) NAMPTCHRM1HTR2AMCHR1MEN1
SCHEMBL882908 0.82 NAMPT (0.46) NAMPTCHRM1HTR2AMCHR1MEN1
SCHEMBL874266 0.81 NAMPT (0.49) NAMPTKITHDAC1CHRM1HTR2A
SCHEMBL3055571 0.80 NAMPT (0.49) NAMPTKITHDAC1CHRM1HTR2A
SCHEMBL882909 0.80 NAMPT (0.49) NAMPTKITHDAC1CHRM1HTR2A
SCHEMBL3055626 0.80 NAMPT (0.48) NAMPTKITHDAC1CHRM1HTR2A
SCHEMBL874907 0.79 NAMPT (0.47) NAMPTKITHDAC1CHRM1HTR2A
SCHEMBL874264 0.79 ALDH1A1 (0.55) MEN1KMT2AALDH1A1
SCHEMBL3050002 0.79 NAMPT (0.47) NAMPTKITHDAC1CHRM1HTR2A
SCHEMBL874755 0.79 NAMPT (0.47) NAMPTKITHDAC1CHRM1HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012038904-A1 NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed
WO-2012038904-A1 NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed