SCHEMBL8760778

SCHEMBL8760778

Brc1ccc(-c2nccc3cc(OCC4CC4CNCC4CC4)ccc23)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LSS P48449 5/20 0.44
SCN9A Q15858 1/20 0.35
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
KDM1A O60341 1/20 0.32
EP300 Q09472 1/20 0.32
AURKA O14965 1/20 0.32
LCK P06239 1/20 0.32
MET P08581 1/20 0.32
KDR P35968 1/20 0.32
TEK Q02763 1/20 0.32
AURKB Q96GD4 1/20 0.32
PDE4A P27815 1/20 0.32
PDE4D Q08499 1/20 0.32
FFAR4 Q5NUL3 1/20 0.32
KHK P50053 1/20 0.31
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31
PARP15 Q460N3 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL8761348 0.93 LSS (0.43) LSSSCN9AAURKALCKMET
SCHEMBL8484710 0.81 LSS (0.55) LSSKDM4E
SCHEMBL8760774 0.80 LSS (0.43) LSSSCN9AKDM4EALDH1A1HPGD
Fumaric Acid SCHEMBL8761342 0.75 LSS (0.42) LSSFFAR4
SCHEMBL8478712 0.75 LSS (0.50) LSSSCN9AKDM1AEP300PARP15
SCHEMBL7687793 0.72 LSS (0.61) LSSALDH1A1MAOBPARP15PARP10
Hydrochloric Acid SCHEMBL7687465 0.71 LSS (0.60) LSSALDH1A1MAOBPARP15PARP10
Fumaric Acid SCHEMBL8484066 0.70 LSS (0.48) LSS
SCHEMBL8484409 0.70 LSS (0.55) LSSKDM4EALDH1A1HPGDMAOA
SCHEMBL8760860 0.69 LSS (0.68) LSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0778271-A2 Aminoalkyl-substituted benzo-heterocyclic compounds F. HOFFMANN-LA ROCHE AG (CH) 1997-06-11 EP claimed
EP-0778271-A2 Aminoalkyl-substituted benzo-heterocyclic compounds F. HOFFMANN-LA ROCHE AG (CH) 1997-06-11 EP disclosed