SCHEMBL8760774

SCHEMBL8760774

NC(CC1CC1COc1ccc2c(-c3ccc(Br)cc3)nccc2c1)C1CC1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
LSS P48449 4/20 0.43
ROCK1 Q13464 1/20 0.31
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
HPGD P15428 1/20 0.30
SCN9A Q15858 1/20 0.30
KDM1A O60341 1/20 0.30
EP300 Q09472 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL8761342 0.92 LSS (0.42) LSS
SCHEMBL8760852 0.80 LSS (0.55) LSSKDM4E
SCHEMBL8478710 0.80 LSS (0.46) LSSROCK1KDM1AEP300
SCHEMBL8760778 0.80 LSS (0.44) LSSKDM4EALDH1A1HPGDSCN9A
Fumaric Acid SCHEMBL8761348 0.74 LSS (0.43) LSSSCN9A
Fumaric Acid SCHEMBL8484063 0.73 LSS (0.44) LSSROCK1
SCHEMBL8478712 0.70 LSS (0.50) LSSROCK1SCN9AKDM1AEP300
SCHEMBL8478588 0.70 LSS (0.66) LSSKDM4E
SCHEMBL8484409 0.69 LSS (0.55) LSSROCK1KDM4EALDH1A1HPGD
SCHEMBL8760860 0.69 LSS (0.68) LSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0778271-A2 Aminoalkyl-substituted benzo-heterocyclic compounds F. HOFFMANN-LA ROCHE AG (CH) 1997-06-11 EP claimed
EP-0778271-A2 Aminoalkyl-substituted benzo-heterocyclic compounds F. HOFFMANN-LA ROCHE AG (CH) 1997-06-11 EP disclosed