SCHEMBL8764371

SCHEMBL8764371

O=C(O)CCC(=O)C(NC(=O)Cn1c(Cc2ccccc2)ccc(NC(=O)CCc2ccccc2)c1=O)SCc1ccccc1Cl

nearest known ligand 0.59

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 10/20 0.59
IL1B P01584 3/20 0.59
ELANE P08246 2/20 0.41
HDAC6 Q9UBN7 2/20 0.37
CTRC Q99895 1/20 0.37
PTGER3 P43115 1/20 0.36
FFAR1 O14842 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
ALOX15 P16050 1/20 0.36
MAPK1 P28482 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12450466 0.84 CASP1 (0.61) CASP1IL1B
SCHEMBL12450470 0.79 CASP1 (0.61) CASP1IL1BELANE
SCHEMBL950212 0.79 CASP1 (0.61) CASP1IL1BELANE
SCHEMBL646080 0.77 CASP1 (0.71) CASP1IL1BELANEMEN1KMT2A
SCHEMBL951210 0.75 CASP1 (0.73) CASP1IL1BELANECTRC
SCHEMBL12914456 0.75 CASP1 (0.62) CASP1IL1B
SCHEMBL645752 0.75 CASP1 (0.62) CASP1IL1B
SCHEMBL12450458 0.75 CASP1 (0.71) CASP1IL1BELANE
SCHEMBL4459947 0.74 CASP1 (1.00) CASP1IL1BELANECTRC
SCHEMBL12522163 0.74 CASP1 (0.83) CASP1IL1BELANECTRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0784628-A1 INHIBITORS OF INTERLEUKIN-1$g(b) CONVERTING ENZYME Vertex Pharmaceuticals Incorporated (US) 1997-07-23 EP disclosed
WO-1995035308-A1 INHIBITORS OF INTERLEUKIN-1β CONVERTING ENZYME VERTEX PHARMACEUTICALS INCORPORATED (US) 1995-12-28 WO disclosed