SCHEMBL8764386

SCHEMBL8764386

NS(=O)(=O)c1ccc(-c2c(-c3ccc(F)cc3)c(C(F)(F)C(F)(F)C(F)(F)F)nn2-c2ccccc2)cc1

nearest known ligand 0.57

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 13/20 0.57
PTGS1 P23219 12/20 0.57
CA1 P00915 4/20 0.46
CA2 P00918 4/20 0.46
CA4 P22748 3/20 0.46
CA9 Q16790 3/20 0.46
PDPK1 O15530 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8765239 0.95 PTGS2 (0.56) PTGS2PTGS1CA1CA2CA4
SCHEMBL8765843 0.94 PTGS2 (0.59) PTGS2PTGS1CA1CA2CA4
SCHEMBL8765792 0.91 PTGS2 (0.48) PTGS2PTGS1
SCHEMBL8635532 0.89 PTGS2 (0.68) PTGS2PTGS1CA1CA2CA4
SCHEMBL8765216 0.88 PTGS2 (0.58) PTGS2PTGS1CA1CA2CA4
SCHEMBL8765041 0.87 PTGS2 (0.59) PTGS2PTGS1CA1CA2CA4
SCHEMBL8631360 0.86 PTGS2 (0.73) PTGS2PTGS1CA1CA2CA4
SCHEMBL8765500 0.85 PTGS2 (0.49) PTGS2PTGS1
SCHEMBL8766115 0.85 PTGS2 (0.54) PTGS2PTGS1
SCHEMBL8764637 0.83 PTGS2 (0.72) PTGS2PTGS1PDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0731794-B1 1,4,5-TRIPHENYL PYRAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION AND INFLAMMATION-RELATED DISORDERS SEARLE & CO (US) 1997-08-06 EP disclosed
EP-0731794-A1 1,4,5-TRIPHENYL PYRAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION AND INFLAMMATION-RELATED DISORDERS SEARLE & CO (US) 1996-09-18 EP disclosed
WO-1995015317-A1 1,4,5-TRIPHENYL PYRAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION AND INFLAMMATION-RELATED DISORDERS G.D. SEARLE & CO. (US) 1995-06-08 WO disclosed