SCHEMBL8764645

SCHEMBL8764645

CC(C)CCNCCCCN1CCCCC1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.48
FPR3 P25089 1/20 0.46
FPR2 P25090 1/20 0.46
SCN5A Q14524 2/20 0.46
MAPT P10636 1/20 0.40
CARM1 Q86X55 1/20 0.39
PRMT6 Q96LA8 1/20 0.39
PRMT8 Q9NR22 1/20 0.39
RAD52 P43351 1/20 0.39
HRH1 P35367 1/20 0.37
TP53 P04637 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
PAOX Q6QHF9 1/20 0.36
SIGMAR1 Q99720 2/20 0.35
KDM1A O60341 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8765083 0.98 HRH3 (0.47) HRH3FPR3FPR2SCN5AMAPT
SCHEMBL9329964 0.95 SCN5A (0.50) HRH3FPR3FPR2SCN5AMAPT
Hydrochloric Acid SCHEMBL9322363 0.93 SCN5A (0.49) HRH3FPR3FPR2SCN5AMAPT
SCHEMBL13519642 0.85 CARM1 (0.50) HRH3FPR3FPR2SCN5ACARM1
SCHEMBL19728165 0.84 SCN5A (0.47) HRH3FPR3FPR2SCN5ACARM1
SCHEMBL29254420 0.82 HRH3 (0.62) HRH3SCN5AMAPTCARM1PRMT6
SCHEMBL441058 0.81 HRH3 (0.61) HRH3FPR3FPR2MAPTHRH1
SCHEMBL10775459 0.80 FPR3 (0.40) HRH3FPR3FPR2SCN5AMAPT
SCHEMBL13160710 0.79 HRH3 (0.54) HRH3FPR3FPR2SCN5ACARM1
SCHEMBL9322157 0.79 HRH3 (0.45) HRH3FPR3FPR2SCN5AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0420116-B1 Novel substituted alkyl piperidines and their use as inhibitors of cholesterol synthesis MERRELL PHARMA INC (US) 1997-07-30 EP claimed
US-5217979-A Substituted alkyl piperidines MERRELL DOW PHARMACEUTICALS INC. (US) 1993-06-08 US claimed
EP-0420116-A2 Novel substituted alkyl piperidines and their use as inhibitors of cholesterol synthesis MERRELL PHARMACEUTICALS INC. (US) 1991-04-03 EP claimed
EP-0420116-B1 Novel substituted alkyl piperidines and their use as inhibitors of cholesterol synthesis MERRELL PHARMA INC (US) 1997-07-30 EP disclosed