SCHEMBL8764845

SCHEMBL8764845

C=CCOC(=O)NC(CC(=O)OCCCC)C(=O)COCc1ccccc1Cl

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 19/20 0.49
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
HPGD P15428 1/20 0.43
CYP2C19 P33261 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1409729 0.85 CASP1 (0.48) CASP1
SCHEMBL7256039 0.85 CASP1 (0.50) CASP1
SCHEMBL646040 0.85 CASP1 (0.65) CASP1
SCHEMBL7345424 0.78 CASP1 (0.44) CASP1HPGD
SCHEMBL8398037 0.75 CASP1 (0.47) CASP1
SCHEMBL4457274 0.75 CASP1 (0.47) CASP1
SCHEMBL12522514 0.74 CASP1 (0.63) CASP1
SCHEMBL949463 0.74 CASP1 (0.63) CASP1
SCHEMBL7005599 0.72 CASP1 (0.43) CASP1
SCHEMBL13139829 0.71 CASP1 (0.50) CASP1CYP1A2CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0784628-A1 INHIBITORS OF INTERLEUKIN-1$g(b) CONVERTING ENZYME Vertex Pharmaceuticals Incorporated (US) 1997-07-23 EP disclosed
WO-1995035308-A1 INHIBITORS OF INTERLEUKIN-1β CONVERTING ENZYME VERTEX PHARMACEUTICALS INCORPORATED (US) 1995-12-28 WO disclosed