SCHEMBL8765208

SCHEMBL8765208

Cc1ccc(-c2c(C(F)(F)F)nn(-c3ccc(C)cc3)c2-c2ccc(S(C)(=O)=O)cc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 18/20 0.60
CYP2C9 P11712 2/20 0.60
PTGS1 P23219 9/20 0.53
CYP2D6 P10635 2/20 0.51
CYP1A2 P05177 1/20 0.51
GRIA2 P42262 1/20 0.51
PDPK1 O15530 2/20 0.47
PTGES O14684 1/20 0.47
HDAC3 O15379 1/20 0.47
CA12 O43570 1/20 0.47
PDE5A O76074 1/20 0.47
ABCB11 O95342 1/20 0.47
MT-CO2 P00403 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
LMNA P02545 1/20 0.47
CA3 P07451 1/20 0.47
CYP3A4 P08684 1/20 0.47
ALOX5 P09917 1/20 0.47
ADORA3 P0DMS8 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8661740 0.95 PTGS2 (0.56) PTGS2CYP2C9PTGS1CYP2D6CYP1A2
SCHEMBL8766098 0.95 CYP1A2 (0.55) PTGS2CYP2C9PTGS1CYP2D6CYP1A2
SCHEMBL8765218 0.94 PTGS2 (0.54) PTGS2CYP2C9PTGS1CYP2D6CYP1A2
SCHEMBL8766070 0.90 PTGS2 (0.60) PTGS2PTGS1CYP2D6CYP1A2GRIA2
SCHEMBL8765162 0.90 PTGS2 (0.62) PTGS2CYP2C9PTGS1CYP2D6CYP1A2
SCHEMBL8765204 0.90 PTGS2 (0.54) PTGS2CYP2C9PTGS1CYP2D6CYP1A2
SCHEMBL8766197 0.89 PTGS2 (0.52) PTGS2CYP2C9PTGS1CYP2D6CYP1A2
SCHEMBL8765415 0.89 PTGS2 (0.67) PTGS2CYP2C9PTGS1CYP2D6PDPK1
SCHEMBL8764563 0.89 PTGS2 (0.55) PTGS2CYP2C9PTGS1CYP2D6CYP1A2
SCHEMBL8765186 0.89 CYP1A2 (0.50) PTGS2CYP2C9PTGS1CYP2D6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0731794-B1 1,4,5-TRIPHENYL PYRAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION AND INFLAMMATION-RELATED DISORDERS SEARLE & CO (US) 1997-08-06 EP disclosed
US-5639777-A 1,4,5-triphenyl pyrazolyl compounds for the treatment of inflammation and inflammation-related disorders G.D. SEARLE & CO. (US) 1997-06-17 US disclosed
US-5401765-A FOR TREATING ARTHRITIS, PAIN AND FEVER Searle, G. D. (US) 1995-03-28 US disclosed