SCHEMBL8765266

SCHEMBL8765266

CS(=O)(=O)c1ccc(-c2c(-c3ccc([N+](=O)[O-])cc3)c(C(F)F)nn2-c2ccc([N+](=O)[O-])cc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 10/20 0.53
PSD A5PKW4 1/20 0.41
MAPT P10636 2/20 0.41
NPC1 O15118 1/20 0.41
ALDH1A1 P00352 1/20 0.41
NFKB1 P19838 1/20 0.41
RAB9A P51151 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
PTGS1 P23219 2/20 0.40
CYP2C9 P11712 1/20 0.40
SRC P12931 1/20 0.40
BRAF P15056 1/20 0.40
KDR P35968 1/20 0.40
CA9 Q16790 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8764581 0.96 PTGS2 (0.49) PTGS2MAPTNPC1ALDH1A1NFKB1
SCHEMBL8765432 0.95 PTGS2 (0.47) PTGS2PSDMAPTNPC1ALDH1A1
SCHEMBL8765507 0.91 PTGS2 (0.43) PTGS2PTGS1CYP2C9
SCHEMBL8765554 0.89 PTGS2 (0.55) PTGS2PTGS1CA9
SCHEMBL8765351 0.86 PTGS2 (0.43) PTGS2PTGS1CYP2C9
SCHEMBL8765305 0.86 PTGS2 (0.51) PTGS2PTGS1CYP2C9
SCHEMBL8765262 0.86 PTGS2 (0.51) PTGS2PTGS1
SCHEMBL8766023 0.85 PTGS2 (0.53) PTGS2MAPTNPC1ALDH1A1NFKB1
SCHEMBL8765498 0.85 PTGS2 (0.51) PTGS2PTGS1
SCHEMBL8765491 0.85 PTGS2 (0.47) PTGS2MAPTNFKB1PTGS1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0731794-B1 1,4,5-TRIPHENYL PYRAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION AND INFLAMMATION-RELATED DISORDERS SEARLE & CO (US) 1997-08-06 EP disclosed
US-5639777-A 1,4,5-triphenyl pyrazolyl compounds for the treatment of inflammation and inflammation-related disorders G.D. SEARLE & CO. (US) 1997-06-17 US disclosed
US-5401765-A FOR TREATING ARTHRITIS, PAIN AND FEVER Searle, G. D. (US) 1995-03-28 US disclosed