SCHEMBL8765747

SCHEMBL8765747

NS(=O)(=O)c1ccc(-c2c(-c3ccc(F)cc3)c(C(F)F)nn2-c2ccc(F)cc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 12/20 0.60
PTGS1 P23219 10/20 0.60
CA1 P00915 6/20 0.53
CA2 P00918 6/20 0.53
CA4 P22748 5/20 0.52
CA9 Q16790 5/20 0.52
CHRNA7 P36544 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8637420 0.94 PTGS2 (0.60) PTGS2PTGS1CA1CA2CA4
SCHEMBL8765925 0.90 PTGS2 (0.51) PTGS2PTGS1CA1CA2CA9
SCHEMBL8764457 0.90 PTGS2 (0.48) PTGS2PTGS1
SCHEMBL8766233 0.89 PTGS2 (0.52) PTGS2PTGS1CA1CA2
SCHEMBL8765145 0.89 PTGS2 (0.60) PTGS2PTGS1CA1CA2CA4
SCHEMBL8765146 0.89 PTGS2 (0.52) PTGS2PTGS1CA1CA2CA4
SCHEMBL8764362 0.89 PTGS2 (0.48) PTGS2PTGS1CA1CA2CA4
SCHEMBL8765285 0.89 PTGS2 (0.60) PTGS2PTGS1CA1CA2CA4
SCHEMBL27459433 0.89 PTGS2 (0.58) PTGS2PTGS1CA1CA2CA9
SCHEMBL8765086 0.88 PTGS2 (0.54) PTGS2PTGS1CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0731794-B1 1,4,5-TRIPHENYL PYRAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION AND INFLAMMATION-RELATED DISORDERS SEARLE & CO (US) 1997-08-06 EP disclosed
US-5639777-A 1,4,5-triphenyl pyrazolyl compounds for the treatment of inflammation and inflammation-related disorders G.D. SEARLE & CO. (US) 1997-06-17 US disclosed
EP-0731794-A1 1,4,5-TRIPHENYL PYRAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION AND INFLAMMATION-RELATED DISORDERS SEARLE & CO (US) 1996-09-18 EP disclosed
WO-1995015317-A1 1,4,5-TRIPHENYL PYRAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION AND INFLAMMATION-RELATED DISORDERS G.D. SEARLE & CO. (US) 1995-06-08 WO disclosed