SCHEMBL8766715

SCHEMBL8766715

C#CC(CCC)(C(=O)O)c1ccco1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.38
HDAC3 O15379 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
HPGD P15428 2/20 0.33
GLA P06280 1/20 0.33
RECQL P46063 1/20 0.33
CYP2C19 P33261 4/20 0.32
ALDH1A1 P00352 4/20 0.32
HTT P42858 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
DPP4 P27487 1/20 0.32
KMT2A Q03164 4/20 0.31
MEN1 O00255 3/20 0.31
TSHR P16473 2/20 0.31
POLB P06746 2/20 0.31
RIPK1 Q13546 1/20 0.31
KDM4E B2RXH2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8765870 0.71 SLC13A5 (0.32) HTT
SCHEMBL8765579 0.71 ESR1 (0.42) MAPTHDAC3HPGDCYP2C19ALDH1A1
SCHEMBL8766524 0.69 CTDSP1 (0.33) CYP2C9
SCHEMBL9402238 0.67 MAPT (0.44) MAPTL3MBTL1RECQLCYP2C19ALDH1A1
SCHEMBL28529969 0.67 KMT2A (0.46) MAPTL3MBTL1RECQLCYP2C19ALDH1A1
SCHEMBL27964089 0.67 MAPT (0.44) MAPTL3MBTL1RECQLCYP2C19ALDH1A1
SCHEMBL5041397 0.65 MAPT (0.43) MAPTL3MBTL1HPGDGLARECQL
Hydrochloric Acid SCHEMBL9402285 0.65 MAPT (0.43) MAPTL3MBTL1RECQLCYP2C19ALDH1A1
SCHEMBL1613425 0.65 MAPT (0.47) MAPTCYP2C19ALDH1A1CYP3A4CYP2D6
SCHEMBL8478567 0.64 PTPN1 (0.42) MAPTL3MBTL1RECQLCYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0785782-A1 DISUBSTITUTED ACETYLENES BEARING HETEROAROMATIC AND HETEROBICYCLIC GROUPS HAVING RETINOID-LIKE ACTIVITY Allergan (US) 1997-07-30 EP disclosed
WO-1996011686-A1 DISUBSTITUTED ACETYLENES BEARING HETEROAROMATIC AND HETEROBICYCLIC GROUPS HAVING RETINOID-LIKE ACTIVITY ALLERGAN (US) 1996-04-25 WO disclosed