SCHEMBL8767124

SCHEMBL8767124

COc1ccc2sc(C(=O)Nc3nnn[nH]3)c(OC(C)C)c2c1.[Na]

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MPO P05164 1/20 0.68
CYSLTR1 Q9Y271 1/20 0.68
ICAM1 P05362 3/20 0.64
SELE P16581 3/20 0.64
VCAM1 P19320 1/20 0.57
EDNRA P25101 1/20 0.44
L3MBTL1 Q9Y468 3/20 0.36
TDP1 Q9NUW8 1/20 0.36
NPC1 O15118 5/20 0.35
RAB9A P51151 5/20 0.35
ALPL P05186 1/20 0.35
ALPI P09923 1/20 0.35
ALPG P10696 1/20 0.35
SMN1; SMN2 Q16637 4/20 0.35
MAPT P10636 3/20 0.35
ALDH1A1 P00352 3/20 0.35
TP53 P04637 1/20 0.35
ALOX15 P16050 1/20 0.35
MAPK1 P28482 1/20 0.35
BACE1 P56817 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6440669 0.99 MPO (0.69) MPOCYSLTR1ICAM1SELEVCAM1
SCHEMBL6568731 0.91 MPO (0.59) MPOCYSLTR1ICAM1SELEVCAM1
SCHEMBL9247114 0.90 MPO (0.56) MPOCYSLTR1ICAM1SELEVCAM1
SCHEMBL9371455 0.89 MPO (0.57) MPOCYSLTR1ICAM1SELEVCAM1
SCHEMBL10372239 0.88 MPO (0.55) MPOCYSLTR1ICAM1SELEVCAM1
SCHEMBL9375225 0.88 ICAM1 (0.57) MPOCYSLTR1ICAM1SELEVCAM1
SCHEMBL10373579 0.87 MPO (0.54) MPOCYSLTR1ICAM1SELEVCAM1
SCHEMBL9246120 0.86 MPO (0.52) MPOCYSLTR1ICAM1SELEVCAM1
SCHEMBL10372978 0.86 MPO (0.52) MPOCYSLTR1ICAM1SELEVCAM1
SCHEMBL9371073 0.86 EDNRA (0.66) MPOCYSLTR1ICAM1SELEVCAM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0789569-A2 USE OF BENZOTHIOPHENES AND BENZOFURANS FOR THE TREATMENT OF INFLAMMATORY BOWEL DISEASE AND INFLAMMATION ASSAY METHOD WARNER-LAMBERT COMPANY (US) 1997-08-20 EP disclosed
WO-1995002406-A2 USE OF BENZOTHIOPHENES AND BENZOFURANS FOR THE TREATMENT OF INFLAMMATORY BOWEL DISEASE AND INFLAMMATION ASSAY METHOD WARNER-LAMBERT COMPANY (US) 1995-01-26 WO disclosed