SCHEMBL8770542

SCHEMBL8770542

CC(C)(C)OC(=O)COc1ccc(N)cc1OCC(=O)OC(C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.45
GAA P10253 2/20 0.45
MAPK1 P28482 1/20 0.43
PTGDR2 Q9Y5Y4 2/20 0.42
KDM4E B2RXH2 3/20 0.42
HPGD P15428 3/20 0.42
HSD17B10 Q99714 2/20 0.42
MEN1 O00255 1/20 0.42
TSHR P16473 1/20 0.42
KMT2A Q03164 1/20 0.42
MAPT P10636 3/20 0.41
POLB P06746 2/20 0.41
CYP2C19 P33261 2/20 0.41
DDB1 Q16531 1/20 0.41
CRBN Q96SW2 1/20 0.41
CYP2C9 P11712 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
ACLY P53396 1/20 0.39
MTNR1A P48039 1/20 0.38
MTNR1B P49286 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1531316 0.93 GAA (0.53) ALDH1A1GAAMAPK1KDM4EMEN1
SCHEMBL13215292 0.88 GAA (0.41) ALDH1A1GAAMAPK1PTGDR2KDM4E
SCHEMBL13623313 0.87 MAPK1 (0.40) ALDH1A1MAPK1PTGDR2KDM4EHPGD
SCHEMBL8770380 0.87 AAK1 (0.40) ALDH1A1MAPK1PTGDR2KDM4EHPGD
SCHEMBL4855128 0.87 MAPK1 (0.51) ALDH1A1GAAMAPK1PTGDR2KDM4E
SCHEMBL13665133 0.83 ALDH1A1 (0.50) ALDH1A1GAAMAPK1KDM4EHPGD
SCHEMBL27539557 0.82 ALDH1A1 (0.48) ALDH1A1MAPK1KDM4EHSD17B10MEN1
Hydrochloric Acid SCHEMBL8474144 0.81 ALDH1A1 (0.51) ALDH1A1GAAMAPK1PTGDR2KDM4E
SCHEMBL7284623 0.80 TSHR (0.51) ALDH1A1GAAMAPK1KDM4EHPGD
SCHEMBL13215511 0.80 PSEN1 (0.38) ALDH1A1GAAMAPK1PTGDR2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0632019-B1 Acylureas ZENECA LTD (GB) 1997-09-24 EP disclosed
US-5576334-A ANTICOAGULANTS ZENECA LIMITED (GB) 1996-11-19 US disclosed
EP-0632019-A1 Acylureas ZENECA LIMITED (GB) 1995-01-04 EP disclosed