SCHEMBL877061

SCHEMBL877061

COCCOc1cc2c(Nc3ccc4c(cnn4C(=O)O)c3)nc(-c3cccc(OCC(=O)NC(C)C)c3)nc2cc1OC

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 11/20 0.54
ROCK1 Q13464 4/20 0.54
CLK2 P49760 1/20 0.54
BLK P51451 1/20 0.54
CSNK2A1 P68400 1/20 0.54
STK3 Q13188 1/20 0.54
DYRK1A Q13627 1/20 0.54
AURKB Q96GD4 1/20 0.54
CLK4 Q9HAZ1 1/20 0.54
STK17A Q9UEE5 1/20 0.54
PRKD3 O94806 1/20 0.45
MET P08581 1/20 0.45
SLC2A1 P11166 7/20 0.44
SLC2A3 P11169 7/20 0.44
ABCB1 P08183 1/20 0.41
ABCG2 Q9UNQ0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3797550 0.92 ROCK2 (0.50) ROCK2ROCK1CLK2BLKCSNK2A1
SCHEMBL4780560 0.89 ERBB2 (0.47) ROCK2ROCK1CLK2BLKCSNK2A1
SCHEMBL878171 0.87 FGFR1 (0.52) ROCK2AURKBPRKD3METABCB1
SCHEMBL877653 0.87 ROCK2 (0.45) ROCK2AURKBPRKD3METABCB1
SCHEMBL877096 0.87 ROCK2 (0.71) ROCK2ROCK1CLK2BLKCSNK2A1
SCHEMBL30915548 0.87 ROCK2 (0.71) ROCK2ROCK1CLK2BLKCSNK2A1
SCHEMBL876538 0.85 ROCK2 (0.74) ROCK2ROCK1CLK2BLKCSNK2A1
SCHEMBL877813 0.84 ABCG2 (0.54) ABCB1ABCG2
SCHEMBL877814 0.84 ABCG2 (0.54) ABCB1ABCG2
SCHEMBL13186724 0.84 ROCK2 (0.47) ROCK2ROCK1CLK2BLKCSNK2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012040499-A2 METABOLIC INHIBITORS SURFACE LOGIX, INC. (US) 2012-03-29 WO disclosed