SCHEMBL8770875

SCHEMBL8770875

COC(=O)CC(O)c1ccc(F)c(F)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.45
CES1 P23141 1/20 0.45
MAPT P10636 3/20 0.44
ALDH1A1 P00352 1/20 0.44
HTT P42858 1/20 0.44
ADRB1 P08588 1/20 0.43
ADRA2A P08913 1/20 0.43
ADRB3 P13945 1/20 0.43
ADRA2B P18089 1/20 0.43
ADRA2C P18825 1/20 0.43
MME P08473 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
PDE4A P27815 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
GAA P10253 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30955364 1.00 CES2 (0.45) CES2CES1MAPTALDH1A1HTT
SCHEMBL20967754 1.00 CES2 (0.45) CES2CES1MAPTALDH1A1HTT
SCHEMBL27932356 0.86 TSHR (0.46) MAPTALDH1A1HTTKDM4EMEN1
SCHEMBL27914160 0.86 TNF (0.43) MAPTALDH1A1HTTL3MBTL1RAB9A
SCHEMBL15189667 0.84 CES2 (0.43) CES2CES1MAPTALDH1A1HTT
SCHEMBL8771004 0.84 CES2 (0.43) CES2CES1MAPTALDH1A1HTT
SCHEMBL8770874 0.83 APP (0.42) CES2CES1ADRB1ADRA2AADRB3
SCHEMBL18898597 0.83 DPP4 (0.47) CES2CES1MAPTALDH1A1HTT
SCHEMBL8770971 0.81 HTT (0.59) MAPTALDH1A1HTTMEN1GAA
SCHEMBL8770905 0.80 CES2 (0.50) CES2CES1MAPTADRB1ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111278809-B Bicyclic sulfones and sulfoxides, and methods of use thereof 豪夫迈·罗氏有限公司 2024-06-25 CN disclosed
EP-3704097-B1 BICYCLIC SULFONES AND SULFOXIDES AND METHODS OF USE THEREOF HOFFMANN LA ROCHE (CH) 2023-10-25 EP disclosed
CN-111278809-A Bicyclic sulfones and sulfoxides, and methods of use thereof 豪夫迈·罗氏有限公司 2020-06-12 CN disclosed
EP-0451668-B1 Process for the production of optically active alkyl 3-aryl-3-hydroxypropionates CHISSO CORP (JP) 1997-08-13 EP disclosed
US-5202457-A Enzyme catalyzed transesterification, resolution of optical active alkyl 3-aryl-3-hydroxypropionate CHISSO CORPORATION (JP) 1993-04-13 US disclosed
EP-0451668-A2 Optically active alkyl 3-aryl-3-hydroxypropionates and a method for producing thereof CHISSO CORPORATION (JP) 1991-10-16 EP disclosed