SCHEMBL8772676

SCHEMBL8772676

C#Cc1c(C(=O)O)cccc1-c1ccc2c(c1)C(=C1CCCCC1)CCC2(C)C

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
RARG P13631 12/20 0.39
RARB P10826 9/20 0.39
RXRA P19793 6/20 0.39
RARA P10276 8/20 0.35
RXRB P28702 3/20 0.32
RXRG P48443 3/20 0.32
P2RX7 Q99572 1/20 0.31
LTB4R2 Q9NPC1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8772694 0.87 RARG (0.42) RARGRARBRXRARARARXRB
SCHEMBL8562392 0.81 RARB (0.42) RARGRARBRXRARARAP2RX7
SCHEMBL8772664 0.76 RARB (0.40) RARGRARBRXRARARA
SCHEMBL8772662 0.74 RARB (0.42) RARGRARBRXRARARA
SCHEMBL8772826 0.72 RARB (0.39) RARGRARBRXRARARALTB4R2
SCHEMBL8772592 0.72 CYP26A1 (0.30) RARGRARBRARA
SCHEMBL8772752 0.72 RARB (0.36) RARGRARBRXRARARA
SCHEMBL8772736 0.72 RARB (0.38) RARGRARBRXRARARA
SCHEMBL8660641 0.71 RARB (0.36) RARGRARBRXRARARALTB4R2
SCHEMBL8836702 0.70 RARB (0.60) RARGRARBRARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0800517-A1 ACETYLENES DISUBSTITUTED WITH A 5 OR 8 SUBSTITUTED TETRAHYDRONAPHTHYL OR DIHYDRONAPHTHYL GROUP AND WITH AN ARYL OR HETEROARYL GROUPS HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY Allergan (US) 1997-10-15 EP disclosed