SCHEMBL8773870

SCHEMBL8773870

CC(=O)Nc1c(F)cc(Br)cc1C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
AKR1C2 P52895 4/20 0.41
AKR1C1 Q04828 4/20 0.41
AKR1C3 P42330 3/20 0.41
AKR1C4 P17516 2/20 0.41
HSD17B10 Q99714 2/20 0.40
MAP2K1 Q02750 1/20 0.39
KDM4E B2RXH2 3/20 0.38
KCNJ11 Q14654 1/20 0.37
HDAC1 Q13547 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
GLA P06280 1/20 0.36
POLB P06746 1/20 0.35
MEN1 O00255 1/20 0.35
MAPK1 P28482 1/20 0.35
KMT2A Q03164 1/20 0.35
DGAT1 O75907 1/20 0.35
NPC1 O15118 1/20 0.35
LMNA P02545 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3726925 0.86 HDAC1 (0.42) ALDH1A1KCNJ11HDAC1HDAC6MEN1
SCHEMBL8528629 0.83 AKR1C3 (0.52) ALDH1A1AKR1C2AKR1C1AKR1C3AKR1C4
SCHEMBL25096707 0.81 ALDH1A1 (0.42) ALDH1A1KCNJ11HDAC1HDAC6MEN1
SCHEMBL3576620 0.80 KDM4E (0.53) ALDH1A1AKR1C2AKR1C1AKR1C3AKR1C4
SCHEMBL3991288 0.80 ALDH1A1 (0.37) ALDH1A1AKR1C2AKR1C1AKR1C3AKR1C4
SCHEMBL4289283 0.79 LCK (0.40) AKR1C2AKR1C1AKR1C3AKR1C4HSD17B10
SCHEMBL30124621 0.78 KMT2A (0.41) ALDH1A1KCNJ11HDAC1HDAC6MEN1
SCHEMBL8773844 0.78 KMT2A (0.41) ALDH1A1KCNJ11HDAC1HDAC6MEN1
SCHEMBL18398288 0.77 KCNJ11 (0.37) ALDH1A1HSD17B10KCNJ11HDAC1HDAC6
SCHEMBL28091550 0.76 KDM4E (0.40) HSD17B10MAP2K1KDM4EHDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0470669-B1 Preparation of fluorophenols, fluorohalophenols, N-acylfluoroanilines, and N-acylfluorohaloanilines DOWELANCO (US) 1997-11-12 EP disclosed
US-5164502-A Fluorinating agents DOWELANCO (US) 1992-11-17 US disclosed
US-5116982-A Fluorination DOWELANCO (US) 1992-05-26 US disclosed
EP-0470669-A2 Preparation of fluorophenols, fluorohalophenols, N-acylfluoroanilines, and N-acylfluorohaloanilines DOWELANCO (US) 1992-02-12 EP disclosed