SCHEMBL8774196

SCHEMBL8774196

CCC1CCC(c2cnc(F)c(F)c2)CC1

nearest known ligand 0.33

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RXRA P19793 5/20 0.33
GRIN1 Q05586 5/20 0.33
GRIN2B Q13224 5/20 0.33
TRPV3 Q8NET8 1/20 0.33
DHODH Q02127 2/20 0.33
ADRB3 P13945 1/20 0.33
ADRA1D P25100 1/20 0.33
SLC6A4 P31645 1/20 0.33
ABAT P80404 1/20 0.33
TMEM97 Q5BJF2 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.31
PDGFRB P09619 1/20 0.31
PDGFRA P16234 1/20 0.31
S1PR1 P21453 1/20 0.30
S1PR3 Q99500 1/20 0.30
PRMT5 O14744 1/20 0.30
PARP1 P09874 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774188 1.00 RXRA (0.33) RXRAGRIN1GRIN2BTRPV3DHODH
SCHEMBL8774166 0.88 CYP2C9 (0.41) RXRAGRIN1GRIN2BDHODHADRB3
SCHEMBL8774158 0.88 CYP2C9 (0.41) RXRAGRIN1GRIN2BDHODHADRB3
SCHEMBL17156238 0.86 KDM4E (0.40) RXRAGRIN1GRIN2BDHODHADRB3
SCHEMBL8774983 0.85 MEN1 (0.37) RXRAGRIN1GRIN2BDHODHADRB3
SCHEMBL8774988 0.85 MEN1 (0.37) RXRAGRIN1GRIN2BDHODHADRB3
SCHEMBL8774474 0.84 CYP2C9 (0.39) RXRAGRIN1GRIN2BDHODHADRB3
SCHEMBL8774438 0.84 MAPT (0.39) RXRAGRIN1GRIN2BDHODHADRB3
SCHEMBL8774494 0.84 CYP2C9 (0.39) RXRAGRIN1GRIN2BDHODHADRB3
SCHEMBL8774484 0.84 CYP2C9 (0.39) RXRAGRIN1GRIN2BDHODHADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed