SCHEMBL8774429

SCHEMBL8774429

CCC1CCC(c2ccc(-c3cc(F)c(F)nc3F)c(F)c2)CC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV3 Q8NET8 1/20 0.36
FASN P49327 1/20 0.32
S1PR4 O95977 1/20 0.31
S1PR1 P21453 1/20 0.31
S1PR5 Q9H228 1/20 0.31
GRM2 Q14416 2/20 0.31
IDO1 P14902 1/20 0.31
KDM5A P29375 1/20 0.30
KDM4C Q9H3R0 1/20 0.30
KDM5B Q9UGL1 1/20 0.30
TLR9 Q9NR96 1/20 0.30
TLR8 Q9NR97 1/20 0.30
TLR7 Q9NYK1 1/20 0.30
DYRK3 O43781 1/20 0.30
PRKD3 O94806 1/20 0.30
MAP4K4 O95819 1/20 0.30
INSR P06213 1/20 0.30
CSF1R P07333 1/20 0.30
PIM1 P11309 1/20 0.30
CLK2 P49760 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774421 1.00 TRPV3 (0.36) TRPV3FASNS1PR4S1PR1S1PR5
SCHEMBL8774806 0.90 CYP2C9 (0.41) TRPV3FASNS1PR4S1PR1S1PR5
SCHEMBL8774680 0.88 MEN1 (0.35)
SCHEMBL8774687 0.88 MEN1 (0.35)
SCHEMBL11115196 0.87 CYP2C9 (0.36) TRPV3FASNKDM5AKDM4CKDM5B
SCHEMBL11115194 0.87 CYP2C9 (0.36) TRPV3FASNKDM5AKDM4CKDM5B
SCHEMBL9160322 0.87 TRPV3 (0.34) TRPV3FASNS1PR4S1PR1S1PR5
SCHEMBL9160310 0.87 TRPV3 (0.34) TRPV3FASNS1PR4S1PR1S1PR5
SCHEMBL8775186 0.87 MAPT (0.37) S1PR1
SCHEMBL8775182 0.87 MAPT (0.37) S1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed