SCHEMBL8774482

SCHEMBL8774482

CCCCc1ccc(-c2ccc(-c3cnc(F)c(F)c3)cc2)c(F)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARB P10826 4/20 0.46
RAB9A P51151 5/20 0.41
SMN1; SMN2 Q16637 5/20 0.41
NPC1 O15118 4/20 0.41
NFKB1 P19838 3/20 0.41
NFKB2 Q00653 3/20 0.41
RELA Q04206 3/20 0.41
MAPK1 P28482 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
RARA P10276 1/20 0.40
RARG P13631 1/20 0.40
S1PR1 P21453 2/20 0.38
S1PR3 Q99500 2/20 0.38
TP53 P04637 2/20 0.38
POLB P06746 1/20 0.38
FDFT1 P37268 1/20 0.37
GAA P10253 2/20 0.37
PSMB5 P28074 1/20 0.37
ALOX5AP P20292 1/20 0.37
FEN1 P39748 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774382 0.96 RARB (0.51) RARBRAB9ASMN1; SMN2NPC1NFKB1
SCHEMBL8774834 0.95 RARB (0.53) RARBRAB9ASMN1; SMN2NPC1L3MBTL1
SCHEMBL8774508 0.95 RARB (0.53) RARBRAB9ASMN1; SMN2NPC1L3MBTL1
SCHEMBL8774684 0.93 RARB (0.43) RARBRAB9ASMN1; SMN2NPC1NFKB1
SCHEMBL8774168 0.92 NPC1 (0.42) RARBRAB9ASMN1; SMN2NPC1S1PR1
SCHEMBL8774371 0.89 RARB (0.48) RARBRAB9ASMN1; SMN2NPC1NFKB1
SCHEMBL8774086 0.89 RARB (0.49) RARBRAB9ASMN1; SMN2NPC1NFKB1
SCHEMBL8774800 0.89 RARB (0.49) RARBRAB9ASMN1; SMN2NPC1NFKB1
SCHEMBL8774727 0.88 RARB (0.50) RARBRAB9ASMN1; SMN2NPC1L3MBTL1
SCHEMBL8774991 0.88 RARB (0.50) RARBRAB9ASMN1; SMN2NPC1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed