SCHEMBL8774588

SCHEMBL8774588

CCOc1ccc(C2CCC(C#Cc3cc(F)c(F)nc3F)CC2)cc1

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 1/20 0.33
MRGPRX4 Q96LA9 1/20 0.32
PGK1 P00558 1/20 0.32
REN P00797 1/20 0.31
CTSD P07339 1/20 0.31
CYP3A4 P08684 1/20 0.31
BACE1 P56817 1/20 0.31
BACE2 Q9Y5Z0 1/20 0.31
SYK P43405 1/20 0.31
NQO1 P15559 1/20 0.31
CACNA2D1 P54289 1/20 0.31
KDM4E B2RXH2 2/20 0.31
ALDH1A1 P00352 2/20 0.31
NPC1 O15118 1/20 0.31
LMNA P02545 1/20 0.31
RAB9A P51151 1/20 0.31
KDM1A O60341 2/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774579 1.00 EGLN1 (0.33) EGLN1MRGPRX4PGK1RENCTSD
SCHEMBL8775115 0.91 RAB9A (0.35) EGLN1MRGPRX4PGK1CYP3A4ALDH1A1
SCHEMBL8775126 0.91 RAB9A (0.35) EGLN1MRGPRX4PGK1CYP3A4ALDH1A1
SCHEMBL8774512 0.91 RAB9A (0.39) EGLN1CYP3A4NPC1LMNARAB9A
SCHEMBL8774525 0.91 RAB9A (0.39) EGLN1CYP3A4NPC1LMNARAB9A
SCHEMBL8774935 0.89 RAB9A (0.38) MRGPRX4CYP3A4LMNARAB9A
SCHEMBL8774930 0.89 RAB9A (0.38) MRGPRX4CYP3A4LMNARAB9A
SCHEMBL8775061 0.89 RAB9A (0.38) LMNARAB9A
SCHEMBL8775065 0.89 RAB9A (0.38) LMNARAB9A
SCHEMBL9153798 0.85 EGLN1 (0.32) EGLN1PGK1NQO1CACNA2D1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed