SCHEMBL8774690

SCHEMBL8774690

CCc1ccc([C@H]2CC[C@H](c3cc(F)c(F)nc3Cl)CC2)cc1

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SOS1 Q07889 2/20 0.34
SPHK1 Q9NYA1 3/20 0.33
DRD2 P14416 1/20 0.32
PANK3 Q9H999 4/20 0.32
LSS P48449 1/20 0.32
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
DGAT1 O75907 1/20 0.31
PDE2A O00408 1/20 0.31
IDO1 P14902 2/20 0.31
AXL P30530 1/20 0.30
ACHE P22303 1/20 0.30
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
KMT2A Q03164 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774697 1.00 SOS1 (0.34) SOS1SPHK1DRD2PANK3LSS
SCHEMBL8774565 0.90 SPHK1 (0.39) SOS1SPHK1DRD2
SCHEMBL8774574 0.90 SPHK1 (0.39) SOS1SPHK1DRD2
SCHEMBL8774560 0.88 SPHK1 (0.35) SPHK1IDO1ALDH1A1MAPT
SCHEMBL8774570 0.88 SPHK1 (0.35) SPHK1IDO1ALDH1A1MAPT
SCHEMBL8774226 0.88 SPHK1 (0.46) SPHK1
SCHEMBL8774234 0.88 SPHK1 (0.46) SPHK1
SCHEMBL8774633 0.87 SPHK1 (0.51) SPHK1
SCHEMBL8774650 0.87 SPHK1 (0.51) SPHK1
SCHEMBL9157415 0.78 SPHK1 (0.34) SPHK1DRD2PANK3LSSCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed