SCHEMBL8776675

SCHEMBL8776675

[O]c1ccc(NC(=O)N2CCN(C3CCNCC3)CC2)cc1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.50
NAMPT P43490 2/20 0.48
CCR2 P41597 4/20 0.47
KCNH2 Q12809 3/20 0.47
CYP2D6 P10635 2/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C19 P33261 1/20 0.46
ALOX5 P09917 1/20 0.45
CYP1A2 P05177 1/20 0.45
MAPT P10636 1/20 0.44
L3MBTL3 Q96JM7 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
FAAH O00519 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8776646 0.89 GAA (0.54) POLBNAMPTCCR2KCNH2CYP2D6
SCHEMBL8776666 0.88 POLB (0.67) POLBNAMPTCCR2CYP2D6CYP3A4
Hydrochloric Acid SCHEMBL9057311 0.84 POLB (0.51) POLBNAMPTCCR2KCNH2CYP2D6
SCHEMBL27498807 0.82 GAA (0.51) POLBNAMPTCCR2KCNH2CYP2D6
SCHEMBL9058915 0.81 MAPT (0.46) POLBCCR2MAPTFAAH
Hydrochloric Acid SCHEMBL9059017 0.80 MAPT (0.45) POLBNAMPTCCR2CYP2D6CYP3A4
SCHEMBL8483552 0.79 POLB (0.45) POLBNAMPTKCNH2CYP2D6CYP1A2
Hydrochloric Acid SCHEMBL9057956 0.78 POLB (0.45) POLBNAMPTCCR2CYP2C19MAPT
Hydrochloric Acid SCHEMBL9058920 0.77 POLB (0.44) POLBNAMPTCCR2KCNH2CYP2D6
SCHEMBL1942072 0.75 CYP3A4 (0.64) CCR2KCNH2CYP2D6CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0799202-A1 PIPERAZINE DERIVATIVES, MEDICAMENTS CONTAINING THE SAME, THEIR USE AND PROCESS FOR PREPARING THE SAME Dr. Karl Thomae GmbH (DE) 1997-10-08 EP disclosed