SCHEMBL8776646

SCHEMBL8776646

O=C(Nc1ccc(O)cc1)N1CCN(C2CCNCC2)CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.54
CA12 O43570 5/20 0.52
CA2 P00918 5/20 0.52
CA9 Q16790 5/20 0.52
CA1 P00915 3/20 0.52
POLB P06746 1/20 0.50
ME2 P23368 1/20 0.49
ME1 P48163 1/20 0.49
ME3 Q16798 1/20 0.49
NAMPT P43490 2/20 0.48
CCR2 P41597 1/20 0.47
KCNH2 Q12809 1/20 0.47
CYP2D6 P10635 2/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C19 P33261 1/20 0.46
ALOX5 P09917 1/20 0.45
CYP1A2 P05177 1/20 0.45
MAPT P10636 1/20 0.44
L3MBTL3 Q96JM7 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27498807 0.92 GAA (0.51) GAACA12CA2CA9CA1
SCHEMBL8776675 0.89 POLB (0.50) POLBNAMPTCCR2KCNH2CYP2D6
SCHEMBL8776666 0.88 POLB (0.67) GAAPOLBNAMPTCCR2CYP2D6
Hydrochloric Acid SCHEMBL9057311 0.84 POLB (0.51) POLBNAMPTCCR2KCNH2CYP2D6
SCHEMBL4391646 0.82 POLB (0.71) GAACA12CA2CA9CA1
SCHEMBL9058915 0.81 MAPT (0.46) POLBCCR2MAPT
SCHEMBL14413284 0.81 CYP3A4 (0.68) GAACA12CA2CA9CA1
Hydrochloric Acid SCHEMBL9059017 0.80 MAPT (0.45) POLBNAMPTCCR2CYP2D6CYP3A4
SCHEMBL27485389 0.79 GAA (0.51) GAACA12CA2CA9CA1
SCHEMBL27484675 0.79 L3MBTL3 (0.64) POLBL3MBTL3L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1183770-A Piperazine derivatives, medicaments containing these compounds, their use and processes for their preparation THOMAE GMBH DR K (DE) 1998-06-03 CN claimed
CN-1183770-A Piperazine derivatives, medicaments containing these compounds, their use and processes for their preparation THOMAE GMBH DR K (DE) 1998-06-03 CN disclosed
EP-0799202-A1 PIPERAZINE DERIVATIVES, MEDICAMENTS CONTAINING THE SAME, THEIR USE AND PROCESS FOR PREPARING THE SAME Dr. Karl Thomae GmbH (DE) 1997-10-08 EP disclosed