SCHEMBL87773

SCHEMBL87773

O=c1cc(-c2ccccc2Cl)oc2ccccc12

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 8/20 0.67
NPC1 O15118 5/20 0.67
RAB9A P51151 4/20 0.67
SMN1; SMN2 Q16637 4/20 0.67
AKR1C3 P42330 1/20 0.67
AKR1C2 P52895 1/20 0.67
AKR1C1 Q04828 1/20 0.67
MEN1 O00255 6/20 0.64
KMT2A Q03164 6/20 0.64
CYP1B1 Q16678 2/20 0.62
CYP1A2 P05177 2/20 0.62
CYP1A1 P04798 1/20 0.62
TNKS O95271 4/20 0.62
CYP3A4 P08684 4/20 0.61
TP53 P04637 3/20 0.61
CYP2C9 P11712 3/20 0.61
CYP2C19 P33261 3/20 0.61
MAPT P10636 3/20 0.61
KDM4E B2RXH2 2/20 0.61
TDP1 Q9NUW8 2/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6907832 0.86 GABRP (0.74) HPGDNPC1RAB9ASMN1; SMN2MEN1
SCHEMBL10810027 0.83 HPGD (0.74) HPGDNPC1RAB9ASMN1; SMN2AKR1C3
SCHEMBL6908632 0.83 GABRP (0.71) HPGDNPC1RAB9ASMN1; SMN2MEN1
SCHEMBL4634256 0.81 HPGD (0.73) HPGDNPC1RAB9ASMN1; SMN2AKR1C3
SCHEMBL25186939 0.80 HPGD (0.67) HPGDNPC1RAB9ASMN1; SMN2AKR1C3
SCHEMBL2436664 0.80 HPGD (0.67) HPGDNPC1RAB9ASMN1; SMN2AKR1C3
SCHEMBL530293 0.80 HPGD (0.67) HPGDNPC1RAB9ASMN1; SMN2AKR1C3
SCHEMBL8025501 0.80 HPGD (0.67) HPGDNPC1RAB9ASMN1; SMN2AKR1C3
SCHEMBL1423180 0.80 HPGD (0.67) HPGDNPC1RAB9ASMN1; SMN2AKR1C3
SCHEMBL312255 0.80 AKR1C3 (1.00) HPGDNPC1RAB9ASMN1; SMN2AKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 370 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025106044-A1 BROMODOMAIN3 (BRD3) INHIBITOR COMPOUND: 4-((4-CHLORO-3-(4-OXO-4 H-CHROMEN-2-YL)PHENYL)SULFONYL)-6-FLUORO-3,4-DIHYDRO-QUINOXAL IN-2(1 H)-ONE T.C. ANKARA UNIVERSITESI REKTORLUGU (TR) 2025-05-22 WO disclosed
CN-119454719-A Application of tripterine as guiding inhibitor of mycobacterium tuberculosis acetyl hydroxy acid synthase 重庆医科大学国际体外诊断研究院 2025-02-18 CN disclosed
CN-118873822-A Treatment of gastrointestinal disorders with TNF inhibitors 比奥拉治疗股份有限公司 2024-11-01 CN disclosed
US-20240224409-A1 ELECTRONIC DEVICE AND MANUFACTURING METHOD THEREOF FUJIFILM CORPORATION (JP) 2024-07-04 US disclosed
US-20240206077-A1 MANUFACTURING METHOD OF ELECTRONIC DEVICE FUJIFILM CORPORATION (JP) 2024-06-20 US disclosed
US-20240196519-A1 ELECTRONIC DEVICE AND MANUFACTURING METHOD THEREOF FUJIFILM CORPORATION (JP) 2024-06-13 US disclosed
US-20240186261-A1 ELECTRONIC DEVICE AND MANUFACTURING METHOD THEREOF FUJIFILM CORPORATION (JP) 2024-06-06 US disclosed
US-20240147630-A1 ELECTRONIC DEVICE AND MANUFACTURING METHOD OF ELECTRONIC DEVICE FUJIFILM CORPORATION (JP) 2024-05-02 US disclosed
WO-2024082757-A1 FLAVONOID COMPOUNDS, GENES ASSOCIATED WITH BIOSYNTHESIS THEREOF AND USE THEREOF 中国科学院青岛生物能源与过程研究所 2024-04-25 WO disclosed
CN-117590691-A Photosensitive resin composition 中央硝子株式会社 2024-02-23 CN disclosed
EP-0860741-B1 Photopolymerizable composition FUJI PHOTO FILM CO LTD (JP) 2001-05-16 EP disclosed
US-6051367-A COMPRISING ONE OR MORE ADDITION-POLYMERIZABLE ETHYLENICALLY UNSATURATED COMPOUNDS AND A SPECIFIC OXIME ETHER COMPOUND; HIGH SENSITIVE TO ACTINIC RAYS RANGING FROM ULTRAVIOLET TO VISIBLE LIGHT, IMPROVED FILM STRENGTH FUJI PHOTO FILM CO., LTD. (JP) 2000-04-18 US disclosed
EP-0973516-A1 USE OF HALO AND/OR NITRO-SUBSTITUTED FLAVONOIDS AS ANXYOLITICS University of Strathclyde (GB) 2000-01-26 EP disclosed
US-5886028-A REDUCING ALCOHOL CONSUMPTION BY ADMINISTERING AN ENZYME INHIBITOR THE ENDOWMENT FOR RESEARCH IN HUMAN BIOLOGY, INC. (US) 1999-03-23 US disclosed
WO-1998044920-A1 USE OF HALO AND/OR NITRO-SUBSTITUTED FLAVONOIDS AS ANXYOLITICS UNIVERSITY OF STRATHCLYDE (GB) 1998-10-15 WO disclosed
EP-0860741-A1 Photopolymerizable composition FUJI PHOTO FILM CO., LTD. (JP) 1998-08-26 EP disclosed
US-5624910-A INHIBITING ALDEHYDE DEHYRDOGENASE ACTIVITY USING DAIDZIN THE ENDOWMENT FOR RESEARCH IN HUMAN BIOLOGY, INC. (US) 1997-04-29 US disclosed
EP-0592583-A1 METHOD FOR THE INHIBITION OF ALDH-I USEFUL IN THE TREATMENT OF ALCOHOL DEPENDENCE OR ALCOHOL ABUSE THE ENDOWMENT FOR RESEARCH IN HUMAN BIOLOGY, INC. (US) 1994-04-20 EP disclosed
US-5204369-A METHOD FOR THE INHIBITION OF ALDH-I USEFUL IN THE TREATMENT OF ALCOHOL DEPENDENCE OR ALCOHOL ABUSE THE ENDOWMENT FOR RESEARCH IN HUMAN BIOLOGY (US) 1993-04-20 US disclosed
WO-1993000896-A1 METHOD FOR THE INHIBITION OF ALDH-I USEFUL IN THE TREATMENT OF ALCOHOL DEPENDENCE OR ALCOHOL ABUSE THE ENDOWMENT FOR RESEARCH IN HUMAN BIOLOGY, INC. (US) 1993-01-21 WO disclosed