SCHEMBL8777350

SCHEMBL8777350

NCCNCCN(C(=O)OCc1ccccc1)C(=O)OCc1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CCR6 P51684 1/20 0.54
PAX8 Q06710 1/20 0.54
HTT P42858 1/20 0.43
ALDH1A1 P00352 3/20 0.42
LMNA P02545 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
MAPK1 P28482 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
SLC6A2 P23975 1/20 0.41
SLC6A3 Q01959 1/20 0.41
KMT2A Q03164 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
CA12 O43570 2/20 0.41
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
CA9 Q16790 2/20 0.41
REN P00797 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5872105 0.88 CCR6 (0.57) CCR6PAX8HTTSMN1; SMN2REN
SCHEMBL1299849 0.88 CCR6 (0.57) CCR6PAX8HTTSMN1; SMN2REN
SCHEMBL10230233 0.86 CCR6 (0.62) CCR6PAX8HTTALDH1A1LMNA
SCHEMBL3372744 0.85 ALDH1A1 (0.50) CCR6PAX8ALDH1A1LMNAMAPK1
SCHEMBL6560598 0.79 HTT (0.54) CCR6PAX8HTTALDH1A1LMNA
SCHEMBL8109244 0.78 ALDH1A1 (0.44) CCR6PAX8ALDH1A1LMNAMAPK1
SCHEMBL17177605 0.78 ALDH1A1 (0.53) HTTALDH1A1LMNASMN1; SMN2MAPK1
SCHEMBL24934482 0.77 CCR6 (0.44) CCR6PAX8ALDH1A1SMN1; SMN2L3MBTL1
SCHEMBL1627692 0.77 ALDH1A1 (0.51) CCR6PAX8HTTALDH1A1LMNA
SCHEMBL15671941 0.77 HTT (0.64) HTTLMNASMN1; SMN2L3MBTL1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0810990-A1 SUBSTITUTED DTPA MONOAMIDES OF CENTRAL CARBOXYLIC ACIDS AND METAL COMPLEXES THEREOF, PHARMACEUTICALS CONTAINING THESE COMPLEXES, DIAGNOSTIC AND THERAPEUTIC USES THEREOF AND METHODS FOR PREPARING THE COMPLEXES AND PHARMACEUTICALS SCHERING AKTIENGESELLSCHAFT (DE) 1997-12-10 EP disclosed
WO-1996026182-A1 SUBSTITUTED DTPA MONOAMIDES OF CENTRAL CARBOXYLIC ACIDS AND METAL COMPLEXES THEREOF, PHARMACEUTICALS CONTAINING THESE COMPLEXES, DIAGNOSTIC AND THERAPEUTIC USES THEREOF AND METHODS FOR PREPARING THE COMPLEXES AND PHARMACEUTICALS SCHERING AKTIENGESELLSCHAFT (DE) 1996-08-29 WO disclosed