SCHEMBL8779946

SCHEMBL8779946

O=[N+]([O-])c1ccc(COP(=O)(CO)OCc2ccc([N+](=O)[O-])cc2)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.71
IDO1 P14902 2/20 0.54
TSHR P16473 1/20 0.51
MAOB P27338 1/20 0.49
PGK1 P00558 1/20 0.48
PGK2 P07205 1/20 0.48
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
ALDH1A1 P00352 3/20 0.46
LOXL2 Q9Y4K0 1/20 0.46
MEN1 O00255 1/20 0.45
POLB P06746 1/20 0.45
KMT2A Q03164 1/20 0.45
CYP2C19 P33261 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CES2 O00748 1/20 0.45
CES1 P23141 1/20 0.45
PLA2G4B P0C869 1/20 0.45
MAPT P10636 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11544092 0.86 AKR1C3 (0.70) AKR1C3IDO1TSHRMAOBPGK1
SCHEMBL5983772 0.83 AKR1C3 (0.81) AKR1C3IDO1TSHRMAOBPGK1
SCHEMBL5069158 0.83 AKR1C3 (1.00) AKR1C3IDO1TSHRMAOBPGK1
SCHEMBL5983768 0.82 AKR1C3 (0.74) AKR1C3IDO1TSHRMAOBPGK1
SCHEMBL8720914 0.80 AKR1C3 (0.60) AKR1C3IDO1TSHRMAOBPGK1
SCHEMBL13537855 0.80 AKR1C3 (0.60) AKR1C3IDO1TSHRNPC1RAB9A
SCHEMBL6932050 0.79 AKR1C3 (0.70) AKR1C3IDO1TSHRMAOBPGK1
SCHEMBL10766432 0.79 AKR1C3 (0.70) AKR1C3IDO1TSHRMAOBPGK1
SCHEMBL5331963 0.78 AKR1C3 (0.67) AKR1C3IDO1TSHRMAOBPGK1
SCHEMBL11655183 0.77 AKR1C3 (0.57) AKR1C3IDO1MAOBPGK1PGK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0539057-B1 Benzimidazole phosphono-amino acids AMERICAN HOME PROD (US) 1997-07-16 EP disclosed
EP-0539057-A1 Benzimidazole phosphono-amino acids AMERICAN HOME PRODUCTS CORPORATION (US) 1993-04-28 EP disclosed
US-5124319-A Administering for treatment of neuropathological disorders induced by overstimulation of excitatory amino acid receptors AMERICAN HOME PRODUCTS CORPORATION (US) 1992-06-23 US disclosed