SCHEMBL8780969

SCHEMBL8780969

OCC[C@]1(c2ccccc2F)CO1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 2/20 0.39
CYP2C9 P11712 1/20 0.39
CYP3A4 P08684 1/20 0.37
HDAC4 P56524 2/20 0.36
BACE1 P56817 3/20 0.34
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
OPRK1 P41145 1/20 0.33
OPRL1 P41146 1/20 0.33
HCAR2 Q8TDS4 1/20 0.32
BACE2 Q9Y5Z0 1/20 0.32
PDK2 Q15119 1/20 0.31
ALDH1A1 P00352 2/20 0.31
USP2 O75604 1/20 0.31
HPGD P15428 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4771886 0.79 HSD11B1 (0.36) HSD11B1CYP2C9CYP3A4
SCHEMBL9005074 0.79 HSD11B1 (0.38) HSD11B1CYP2C9CYP3A4BACE1HCAR2
SCHEMBL3454385 0.79 HSD11B1 (0.36) HSD11B1CYP2C9CYP3A4
SCHEMBL8723263 0.79 HSD11B1 (0.38) HSD11B1CYP2C9CYP3A4BACE1HCAR2
SCHEMBL18754946 0.74 PDE2A (0.37)
SCHEMBL2874324 0.73 HSD11B1 (0.37) HSD11B1CYP2C9OPRM1OPRL1
SCHEMBL28721499 0.72 KMT2A (0.36) ALDH1A1HPGD
SCHEMBL23612354 0.69 HDAC4 (0.37) HDAC4BACE1OPRM1OPRD1OPRK1
SCHEMBL15705147 0.68 BACE1 (0.33) HDAC4BACE1HCAR2
SCHEMBL17673207 0.67 BACE1 (0.40) HDAC4BACE1HCAR2BACE2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0809640-A1 AZOLE COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-12-03 EP disclosed
WO-1996025410-A1 AZOLE COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-08-22 WO disclosed